Taselisib KINOMEscan - Dataset (ID:20264)

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Small Molecule Protein % Control Assay compound conc Conc unit
Taselisib MTOR 90.0 100
nM
Taselisib FLT3(ITD,D835V) 90.0 100
nM
Taselisib ABL1(F317L)-nonphosphorylated 90.0 100
nM
Taselisib FGR 90.0 1000
nM
Taselisib SRC 90.0 100
nM
Taselisib ANKK1 90.0 100
nM
Taselisib EGFR(T790M) 90.0 100
nM
Taselisib MAP3K1 90.0 100
nM
Taselisib ABL1-phosphorylated 91.0 100
nM
Taselisib EGFR(L747-S752del, P753S) 91.0 1000
nM
Taselisib LOK 91.0 100
nM
Taselisib KPCI 91.0 1000
nM
Taselisib KGP1 91.0 1000
nM
Taselisib DCAMKL3 91.0 100
nM
Taselisib RSK4(Kin.Dom.1-N-terminal) 91.0 100
nM
Taselisib DAPK2 91.0 100
nM
Taselisib MARK1 91.0 1000
nM
Taselisib RSK3(Kin.Dom.2-C-terminal) 91.0 1000
nM
Taselisib TIE2 91.0 100
nM
Taselisib HIPK4 91.0 100
nM
Taselisib BRAF 91.0 1000
nM
Taselisib CLK3 91.0 100
nM
Taselisib BMPR1B 91.0 100
nM
Taselisib GRK7 91.0 100
nM
Taselisib IGF1R 91.0 100
nM