Taselisib KINOMEscan - Dataset (ID:20264)
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Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
Taselisib | AMPK-alpha2 | 89.0 | 100 | nM |
Taselisib | EGFR(L858R,T790M) | 69.0 | 100 | nM |
Taselisib | CAMKK2 | 85.0 | 100 | nM |
Taselisib | EGFR(L861Q) | 95.0 | 100 | nM |
Taselisib | AAK1 | 77.0 | 100 | nM |
Taselisib | EGFR(S752-I759del) | 93.0 | 100 | nM |
Taselisib | CASK | 75.0 | 100 | nM |
Taselisib | EGFR(T790M) | 90.0 | 100 | nM |
Taselisib | ANKK1 | 90.0 | 100 | nM |
Taselisib | EIF2AK1 | 96.0 | 100 | nM |
Taselisib | CDC2L1 | 100.0 | 100 | nM |
Taselisib | EPHA1 | 100.0 | 100 | nM |
Taselisib | ABL2 | 94.0 | 100 | nM |
Taselisib | EPHA2 | 80.0 | 100 | nM |
Taselisib | CDC2L2 | 100.0 | 100 | nM |
Taselisib | EPHA3 | 94.0 | 100 | nM |
Taselisib | NUAK1 | 97.0 | 100 | nM |
Taselisib | EPHA4 | 94.0 | 100 | nM |
Taselisib | CDC2L5 | 81.0 | 100 | nM |
Taselisib | EPHA5 | 96.0 | 100 | nM |
Taselisib | ABL1(M351T)-phosphorylated | 94.0 | 100 | nM |
Taselisib | EPHA6 | 95.0 | 100 | nM |
Taselisib | CDK11 | 76.0 | 100 | nM |
Taselisib | EPHA7 | 98.0 | 100 | nM |
Taselisib | MST2 | 100.0 | 100 | nM |