Taselisib KINOMEscan - Dataset (ID:20264)

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Small Molecule Protein % Control Assay compound conc Conc unit
Taselisib AMPK-alpha2 89.0 100
nM
Taselisib EGFR(L858R,T790M) 69.0 100
nM
Taselisib CAMKK2 85.0 100
nM
Taselisib EGFR(L861Q) 95.0 100
nM
Taselisib AAK1 77.0 100
nM
Taselisib EGFR(S752-I759del) 93.0 100
nM
Taselisib CASK 75.0 100
nM
Taselisib EGFR(T790M) 90.0 100
nM
Taselisib ANKK1 90.0 100
nM
Taselisib EIF2AK1 96.0 100
nM
Taselisib CDC2L1 100.0 100
nM
Taselisib EPHA1 100.0 100
nM
Taselisib ABL2 94.0 100
nM
Taselisib EPHA2 80.0 100
nM
Taselisib CDC2L2 100.0 100
nM
Taselisib EPHA3 94.0 100
nM
Taselisib NUAK1 97.0 100
nM
Taselisib EPHA4 94.0 100
nM
Taselisib CDC2L5 81.0 100
nM
Taselisib EPHA5 96.0 100
nM
Taselisib ABL1(M351T)-phosphorylated 94.0 100
nM
Taselisib EPHA6 95.0 100
nM
Taselisib CDK11 76.0 100
nM
Taselisib EPHA7 98.0 100
nM
Taselisib MST2 100.0 100
nM