Taselisib KINOMEscan - Dataset (ID:20264)
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Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
Taselisib | DRAK1 | 100.0 | 100 | nM |
Taselisib | ALK(C1156Y) | 79.0 | 100 | nM |
Taselisib | DRAK2 | 94.0 | 100 | nM |
Taselisib | CAMK2A | 95.0 | 100 | nM |
Taselisib | DYRK1A | 83.0 | 100 | nM |
Taselisib | ABL1-nonphosphorylated | 88.0 | 100 | nM |
Taselisib | DYRK1B | 74.0 | 100 | nM |
Taselisib | CAMK2B | 93.0 | 100 | nM |
Taselisib | DYRK2 | 93.0 | 100 | nM |
Taselisib | ALK(L1196M) | 78.0 | 100 | nM |
Taselisib | EGFR | 96.0 | 100 | nM |
Taselisib | KCC2D | 84.0 | 100 | nM |
Taselisib | EGFR(E746-A750del) | 89.0 | 100 | nM |
Taselisib | ABL1(H396P)-phosphorylated | 80.0 | 100 | nM |
Taselisib | EGFR(G719C) | 93.0 | 100 | nM |
Taselisib | CAMK2G | 92.0 | 100 | nM |
Taselisib | EGFR(G719S) | 98.0 | 100 | nM |
Taselisib | AMPK-alpha1 | 93.0 | 100 | nM |
Taselisib | EGFR(L747-E749del, A750P) | 100.0 | 100 | nM |
Taselisib | KCC4 | 75.0 | 100 | nM |
Taselisib | EGFR(L747-S752del, P753S) | 88.0 | 100 | nM |
Taselisib | ABL1-phosphorylated | 91.0 | 100 | nM |
Taselisib | EGFR(L747-T751del,Sins) | 88.0 | 100 | nM |
Taselisib | KKCC1 | 96.0 | 100 | nM |
Taselisib | MARK4 | 100.0 | 100 | nM |