Taselisib KINOMEscan - Dataset (ID:20264)

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Small Molecule Protein % Control Assay compound conc Conc unit
Taselisib DRAK1 100.0 100
nM
Taselisib ALK(C1156Y) 79.0 100
nM
Taselisib DRAK2 94.0 100
nM
Taselisib CAMK2A 95.0 100
nM
Taselisib DYRK1A 83.0 100
nM
Taselisib ABL1-nonphosphorylated 88.0 100
nM
Taselisib DYRK1B 74.0 100
nM
Taselisib CAMK2B 93.0 100
nM
Taselisib DYRK2 93.0 100
nM
Taselisib ALK(L1196M) 78.0 100
nM
Taselisib EGFR 96.0 100
nM
Taselisib KCC2D 84.0 100
nM
Taselisib EGFR(E746-A750del) 89.0 100
nM
Taselisib ABL1(H396P)-phosphorylated 80.0 100
nM
Taselisib EGFR(G719C) 93.0 100
nM
Taselisib CAMK2G 92.0 100
nM
Taselisib EGFR(G719S) 98.0 100
nM
Taselisib AMPK-alpha1 93.0 100
nM
Taselisib EGFR(L747-E749del, A750P) 100.0 100
nM
Taselisib KCC4 75.0 100
nM
Taselisib EGFR(L747-S752del, P753S) 88.0 100
nM
Taselisib ABL1-phosphorylated 91.0 100
nM
Taselisib EGFR(L747-T751del,Sins) 88.0 100
nM
Taselisib KKCC1 96.0 100
nM
Taselisib MARK4 100.0 100
nM