Taselisib KINOMEscan - Dataset (ID:20264)

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Small Molecule Protein % Control Assay compound conc Conc unit
Taselisib ABL1(F317I)-nonphosphorylated 100.0 1000
nM
Taselisib ABL1(Y253F)-phosphorylated 100.0 1000
nM
Taselisib AURKB 100.0 1000
nM
Taselisib NUAK1 100.0 1000
nM
Taselisib ABL1(T315I)-phosphorylated 100.0 100
nM
Taselisib ABL1-phosphorylated 100.0 1000
nM
Taselisib ABL1(H396P)-phosphorylated 100.0 1000
nM
Taselisib ABL2 100.0 1000
nM
Taselisib ACVR1 100.0 100
nM
Taselisib ACVR1 100.0 1000
nM
Taselisib ABL1(M351T)-phosphorylated 100.0 1000
nM
Taselisib BLK 100.0 1000
nM
Taselisib BMPR1A 100.0 100
nM
Taselisib BMX 100.0 1000
nM
Taselisib BRSK1 100.0 100
nM
Taselisib ALK 100.0 1000
nM
Taselisib ACVRL1 100.0 100
nM
Taselisib ACVRL1 100.0 1000
nM
Taselisib ADCK3 100.0 100
nM
Taselisib ADCK3 100.0 1000
nM
Taselisib ADCK4 100.0 100
nM
Taselisib ADCK4 100.0 1000
nM
Taselisib ABL1(T315I)-nonphosphorylated 100.0 1000
nM
Taselisib CDK2 100.0 1000
nM
Taselisib CDK11 100.0 1000
nM