Taselisib KINOMEscan - Dataset (ID:20264)

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Small Molecule Protein % Control Assay compound conc Conc unit
Taselisib EGFR(L858R) 90.0 1000
nM
Taselisib KKCC1 100.0 1000
nM
Taselisib EGFR(L858R,T790M) 98.0 1000
nM
Taselisib MLK1 92.0 1000
nM
Taselisib EGFR(L861Q) 79.0 1000
nM
Taselisib CAMKK2 96.0 1000
nM
Taselisib EGFR(S752-I759del) 99.0 1000
nM
Taselisib AMPK-alpha2 99.0 1000
nM
Taselisib EGFR(T790M) 100.0 1000
nM
Taselisib CASK 76.0 1000
nM
Taselisib EIF2AK1 100.0 1000
nM
Taselisib ABL1-phosphorylated 100.0 1000
nM
Taselisib EPHA1 100.0 1000
nM
Taselisib CDC2L1 100.0 1000
nM
Taselisib EPHA2 100.0 1000
nM
Taselisib ANKK1 89.0 1000
nM
Taselisib EPHA3 98.0 1000
nM
Taselisib CDC2L2 100.0 1000
nM
Taselisib EPHA4 95.0 1000
nM
Taselisib ABL1(H396P)-phosphorylated 100.0 1000
nM
Taselisib EPHA5 95.0 1000
nM
Taselisib CDC2L5 91.0 1000
nM
Taselisib EPHA6 92.0 1000
nM
Taselisib NUAK1 100.0 1000
nM
Taselisib MST2 98.0 1000
nM