Taselisib KINOMEscan - Dataset (ID:20264)

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Small Molecule Protein % Control Assay compound conc Conc unit
Taselisib ABL1(T315I)-phosphorylated 100.0 1000
nM
Taselisib ABL1(Y253F)-phosphorylated 96.0 100
nM
Taselisib ABL1(Y253F)-phosphorylated 100.0 1000
nM
Taselisib ABL1-nonphosphorylated 88.0 100
nM
Taselisib ABL1-nonphosphorylated 97.0 1000
nM
Taselisib ABL1-phosphorylated 91.0 100
nM
Taselisib ABL1-phosphorylated 100.0 1000
nM
Taselisib ABL2 94.0 100
nM
Taselisib ABL2 100.0 1000
nM
Taselisib ACVR1 100.0 100
nM
Taselisib ACVR1 100.0 1000
nM
Taselisib ACVR1B 99.0 100
nM
Taselisib ACVR1B 97.0 1000
nM
Taselisib ACVR2A 99.0 100
nM
Taselisib ACVR2A 97.0 1000
nM
Taselisib ACVR2B 92.0 100
nM
Taselisib ACVR2B 92.0 1000
nM
Taselisib ACVRL1 100.0 100
nM
Taselisib ACVRL1 100.0 1000
nM
Taselisib ADCK3 100.0 100
nM
Taselisib ADCK3 100.0 1000
nM
Taselisib ADCK4 100.0 100
nM
Taselisib ADCK4 100.0 1000
nM
Taselisib AKT1 92.0 100
nM
Taselisib AKT1 100.0 1000
nM