GDC-0941 KINOMEscan-3 - Dataset (ID:20261)

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Small Molecule Protein % Control Assay compound conc Conc unit
Pictilisib ACVR1B 100.0 1000
nM
Pictilisib ADCK4 87.0 1000
nM
Pictilisib ABL1-nonphosphorylated 85.0 1000
nM
Pictilisib ACVR1 100.0 1000
nM
Pictilisib ACVR2B 100.0 1000
nM
Pictilisib ADCK3 91.0 1000
nM
Pictilisib ABL1(T315I)-phosphorylated 100.0 1000
nM
Pictilisib ABL1(Y253F)-phosphorylated 100.0 1000
nM
Pictilisib ABL1-phosphorylated 99.0 1000
nM
Pictilisib ABL2 99.0 1000
nM
Pictilisib ACVR2A 88.0 1000
nM
Pictilisib ABL1(F317I)-nonphosphorylated 100.0 1000
nM
Pictilisib ABL1(H396P)-nonphosphorylated 81.0 1000
nM
Pictilisib ACVRL1 100.0 1000
nM
Pictilisib ABL1(H396P)-phosphorylated 100.0 1000
nM
Pictilisib ABL1(F317I)-phosphorylated 100.0 1000
nM
Pictilisib ABL1(M351T)-phosphorylated 100.0 1000
nM
Pictilisib ABL1(E255K)-phosphorylated 85.0 1000
nM
Pictilisib ABL1(Q252H)-nonphosphorylated 80.0 1000
nM
Pictilisib ABL1(F317L)-nonphosphorylated 100.0 1000
nM
Pictilisib ABL1(Q252H)-phosphorylated 100.0 1000
nM
Pictilisib AAK1 93.0 1000
nM
Pictilisib ABL1(T315I)-nonphosphorylated 96.0 1000
nM
Pictilisib ABL1(F317L)-phosphorylated 100.0 1000
nM
Pictilisib AKT1 100.0 1000
nM
  • Page 1 of 38
  • 1 to 25 of 936 records