GDC-0941 KINOMEscan-3 - Dataset (ID:20261)

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Small Molecule Protein % Control Assay compound conc Conc unit
Pictilisib PIK3CA(E545A) 0.0 1000
nM
Pictilisib PIK3CA(E542K) 0.0 1000
nM
Pictilisib PIK3CA(H1047Y) 0.0 1000
nM
Pictilisib PIK3CA(C420R) 0.0 1000
nM
Pictilisib PIK3CA(I800L) 0.0 1000
nM
Pictilisib PIK3CB 0.0 1000
nM
Pictilisib PIK3CA(M1043I) 0.0 100
nM
Pictilisib PIK3CD 0.0 1000
nM
Pictilisib PIK3CA(E545K) 0.0 1000
nM
Pictilisib PIK3CA(Q546K) 0.1 1000
nM
Pictilisib PIK3CA 0.2 1000
nM
Pictilisib PIK3CA(M1043I) 0.4 1000
nM
Pictilisib PIK3CA(E545K) 0.8 100
nM
Pictilisib PIK3CA(H1047L) 0.8 1000
nM
Pictilisib PIK3CA(H1047Y) 1.0 100
nM
Pictilisib PIK3CA(E542K) 1.2 100
nM
Pictilisib PIK3CA(E545A) 1.6 100
nM
Pictilisib PIK3CA(C420R) 1.9 100
nM
Pictilisib PIK3CG 3.5 1000
nM
Pictilisib PIK3CA 3.5 100
nM
Pictilisib PIK3CA(Q546K) 4.0 100
nM
Pictilisib FYV1 4.5 1000
nM
Pictilisib PIK3CA(I800L) 7.0 100
nM
Pictilisib PIK3CD 7.0 100
nM
Pictilisib MTOR 13.0 1000
nM
  • Page 1 of 38
  • 1 to 25 of 936 records