5z-7-oxozeaenol KiNativ -- single dose experiment - Dataset (ID:20255)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
5z-7-oxozeaenol | MWCL.1 | NEK7 | AACLLDGVPVALKK | Lys1 | 25.7 | 1 | uM |
5z-7-oxozeaenol | MWCL.1 | NEK8 | DLKTQNILLDK | Lys2 | -7.9 | 1 | uM |
5z-7-oxozeaenol | MWCL.1 | NEK9 | DIKTLNIFLTK | Lys2 | -37.5 | 1 | uM |
5z-7-oxozeaenol | MWCL.1 | OSR1 | DVKAGNILLGEDGSVQIADFGVSAFLATGGDITR | Lys2 | 6.2 | 1 | uM |
5z-7-oxozeaenol | MWCL.1 | p38a | DLKPSNLAVNEDCELK | Lys2 | 6.3 | 1 | uM |
5z-7-oxozeaenol | MWCL.1 | p38d,p38g | DLKPGNLAVNEDCELK | Lys2 | -1.4 | 1 | uM |
5z-7-oxozeaenol | MWCL.1 | PAN3 | VMDPTKILITGK | ATP | 17.1 | 1 | uM |
5z-7-oxozeaenol | MWCL.1 | PCTAIRE2,PCTAIRE3 | SKLTENLVALKEIR | Lys1 | -31.2 | 1 | uM |
5z-7-oxozeaenol | MWCL.1 | PDHK1 | SPGQPIQVVYVPSHLYHMVFELFKNAMR | Other | -26.7 | 1 | uM |
5z-7-oxozeaenol | MWCL.1 | PDK1 | EYAIKILEK | Lys1 | 1 | uM | |
5z-7-oxozeaenol | MWCL.1 | PEK | DLKPSNIFFTMDDVVK | Lys2 | 39.8 | 1 | uM |
5z-7-oxozeaenol | MWCL.1 | PHKg1 | DLKPENILLDDNMNIK | Lys2 | -11.8 | 1 | uM |
5z-7-oxozeaenol | MWCL.1 | PHKg2 | ATGHEFAVKIMEVTAER | Lys1 | 1 | uM | |
5z-7-oxozeaenol | MWCL.1 | PI4KA,PI4KAP2 | SGTPMQSAAKAPYLAK | ATP | 46.0 | 1 | uM |
5z-7-oxozeaenol | MWCL.1 | PI4KB | VPHTQAVVLNSKDK | ATP | -10.4 | 1 | uM |
5z-7-oxozeaenol | MWCL.1 | PIK3C2B | VIFKCGDDLRQDMLTLQMIR | ATP | 1 | uM | |
5z-7-oxozeaenol | MWCL.1 | PIK3C3 | TEDGGKYPVIFKHGDDLR | ATP | -38.5 | 1 | uM |
5z-7-oxozeaenol | MWCL.1 | PIK3CB | VFGEDSVGVIFKNGDDLRQDMLTLQMLR | ATP | 17.3 | 1 | uM |
5z-7-oxozeaenol | MWCL.1 | PIK3CD | VNWLAHNVSKDNRQ | ATP | -0.3 | 1 | uM |
5z-7-oxozeaenol | MWCL.1 | PIK3CG | KKPLWLEFK | ATP | 36.0 | 1 | uM |
5z-7-oxozeaenol | MWCL.1 | PIP4K2A | AKELPTLKDNDFINEGQK | ATP | 7.1 | 1 | uM |
5z-7-oxozeaenol | MWCL.1 | FYV1 | GGKSGAAFYATEDDRFILK | ATP | 4.8 | 1 | uM |
5z-7-oxozeaenol | MWCL.1 | PITSLRE | DLKTSNLLLSHAGILK | Lys2 | 1.3 | 1 | uM |
5z-7-oxozeaenol | MWCL.1 | PKD2 | DVAVKVIDK | Lys1 | 11.9 | 1 | uM |
5z-7-oxozeaenol | MWCL.1 | PKD3 | DVAIKVIDK | Lys1 | -16.0 | 1 | uM |