5z-7-oxozeaenol KiNativ -- single dose experiment - Dataset (ID:20255)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
5z-7-oxozeaenol MWCL.1 CaMK2g
TSTQEYAAKIINTK
Lys1
-3.8
1
uM
5z-7-oxozeaenol MWCL.1 CaMKK2
DIKPSNLLVGEDGHIK
Lys2
-16.3
1
uM
5z-7-oxozeaenol BCWM.1 CaMKK2
DIKPSNLLVGEDGHIK
Lys2
8.9
1
uM
5z-7-oxozeaenol BCWM.1 CASK
ETGQQFAVKIVDVAK
Lys1
-20.9
1
uM
5z-7-oxozeaenol MWCL.1 CASK
ETGQQFAVKIVDVAK
Lys1
-22.6
1
uM
5z-7-oxozeaenol MWCL.1 CDC2
DLKPQNLLIDDKGTIK
Lys2
-2.5
1
uM
5z-7-oxozeaenol BCWM.1 CDC2
DLKPQNLLIDDKGTIK
Lys2
9.4
1
uM
5z-7-oxozeaenol MWCL.1 CDK11,CDK8
DLKPANILVMGEGPER
Lys2
37.2
1
uM
5z-7-oxozeaenol BCWM.1 CDK11,CDK8
DLKPANILVMGEGPER
Lys2
7.7
1
uM
5z-7-oxozeaenol MWCL.1 CDK14
LVALKVIR
Lys1
-17.9
1
uM
5z-7-oxozeaenol BCWM.1 CDK14
LVALKVIR
Lys1
7.5
1
uM
5z-7-oxozeaenol MWCL.1 CDK16
SKLTDNLVALKEIR
Lys1
1
uM
5z-7-oxozeaenol BCWM.1 CDK16
SKLTDNLVALKEIR
Lys1
-10.8
1
uM
5z-7-oxozeaenol MWCL.1 CDK2
DLKPQNLLINTEGAIK
Lys2
-9.2
1
uM
5z-7-oxozeaenol BCWM.1 CDK2
DLKPQNLLINTEGAIK
Lys2
5.0
1
uM
5z-7-oxozeaenol MWCL.1 CDK4
DLKPENILVTSGGTVK
Lys2
9.7
1
uM
5z-7-oxozeaenol BCWM.1 CDK4
DLKPENILVTSGGTVK
Lys2
21.8
1
uM
5z-7-oxozeaenol MWCL.1 CDK5
DLKPQNLLINR
Lys2
-4.2
1
uM
5z-7-oxozeaenol BCWM.1 CDK5
DLKPQNLLINR
Lys2
9.6
1
uM
5z-7-oxozeaenol MWCL.1 CDK6
DLKPQNILVTSSGQIK
Lys2
1.2
1
uM
5z-7-oxozeaenol BCWM.1 CDK6
DLKPQNILVTSSGQIK
Lys2
10.3
1
uM
5z-7-oxozeaenol MWCL.1 CDK7
DLKPNNLLLDENGVLK
Lys2
-30.3
1
uM
5z-7-oxozeaenol BCWM.1 CDK7
DLKPNNLLLDENGVLK
Lys2
-3.8
1
uM
5z-7-oxozeaenol MWCL.1 CDK9
DMKAANVLITR
Lys2
25.9
1
uM
5z-7-oxozeaenol BCWM.1 CDK9
DMKAANVLITR
Lys2
25.0
1
uM