5z-7-oxozeaenol KiNativ -- single dose experiment - Dataset (ID:20255)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
5z-7-oxozeaenol | MWCL.1 | CaMK2g | TSTQEYAAKIINTK | Lys1 | -3.8 | 1 | uM |
5z-7-oxozeaenol | MWCL.1 | CaMKK2 | DIKPSNLLVGEDGHIK | Lys2 | -16.3 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | CaMKK2 | DIKPSNLLVGEDGHIK | Lys2 | 8.9 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | CASK | ETGQQFAVKIVDVAK | Lys1 | -20.9 | 1 | uM |
5z-7-oxozeaenol | MWCL.1 | CASK | ETGQQFAVKIVDVAK | Lys1 | -22.6 | 1 | uM |
5z-7-oxozeaenol | MWCL.1 | CDC2 | DLKPQNLLIDDKGTIK | Lys2 | -2.5 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | CDC2 | DLKPQNLLIDDKGTIK | Lys2 | 9.4 | 1 | uM |
5z-7-oxozeaenol | MWCL.1 | CDK11,CDK8 | DLKPANILVMGEGPER | Lys2 | 37.2 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | CDK11,CDK8 | DLKPANILVMGEGPER | Lys2 | 7.7 | 1 | uM |
5z-7-oxozeaenol | MWCL.1 | CDK14 | LVALKVIR | Lys1 | -17.9 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | CDK14 | LVALKVIR | Lys1 | 7.5 | 1 | uM |
5z-7-oxozeaenol | MWCL.1 | CDK16 | SKLTDNLVALKEIR | Lys1 | 1 | uM | |
5z-7-oxozeaenol | BCWM.1 | CDK16 | SKLTDNLVALKEIR | Lys1 | -10.8 | 1 | uM |
5z-7-oxozeaenol | MWCL.1 | CDK2 | DLKPQNLLINTEGAIK | Lys2 | -9.2 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | CDK2 | DLKPQNLLINTEGAIK | Lys2 | 5.0 | 1 | uM |
5z-7-oxozeaenol | MWCL.1 | CDK4 | DLKPENILVTSGGTVK | Lys2 | 9.7 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | CDK4 | DLKPENILVTSGGTVK | Lys2 | 21.8 | 1 | uM |
5z-7-oxozeaenol | MWCL.1 | CDK5 | DLKPQNLLINR | Lys2 | -4.2 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | CDK5 | DLKPQNLLINR | Lys2 | 9.6 | 1 | uM |
5z-7-oxozeaenol | MWCL.1 | CDK6 | DLKPQNILVTSSGQIK | Lys2 | 1.2 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | CDK6 | DLKPQNILVTSSGQIK | Lys2 | 10.3 | 1 | uM |
5z-7-oxozeaenol | MWCL.1 | CDK7 | DLKPNNLLLDENGVLK | Lys2 | -30.3 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | CDK7 | DLKPNNLLLDENGVLK | Lys2 | -3.8 | 1 | uM |
5z-7-oxozeaenol | MWCL.1 | CDK9 | DMKAANVLITR | Lys2 | 25.9 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | CDK9 | DMKAANVLITR | Lys2 | 25.0 | 1 | uM |