5z-7-oxozeaenol KiNativ -- single dose experiment - Dataset (ID:20255)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
5z-7-oxozeaenol MWCL.1 MK01
DLKPSNLLLNTTCDLK
Lys2
1.1
1
uM
5z-7-oxozeaenol MWCL.1 MST1
ETGQIVAIKQVPVESDLQEIIK
Lys1
-11.0
1
uM
5z-7-oxozeaenol BCWM.1 LATS2
DIKPDNILIDLDGHIK
Lys2
-11.0
1
uM
5z-7-oxozeaenol BCWM.1 GCN2_domain2
DLKPVNIFLDSDDHVK
Lys2
11.0
1
uM
5z-7-oxozeaenol BCWM.1 CAMK1D
LFAVKCIPK
Lys1
11.1
1
uM
5z-7-oxozeaenol BCWM.1 RIPK2
VQVAVKHLHIHTPLLDSER
Lys1
11.1
1
uM
5z-7-oxozeaenol BCWM.1 TYK2(Kin.Dom.2)
IGDFGLAKAVPEGHEYYR
Activation Loop
11.1
1
uM
5z-7-oxozeaenol BCWM.1 SNRK
DLKPENVVFFEK
Lys2
-11.3
1
uM
5z-7-oxozeaenol BCWM.1 M4K3
NVNTGELAAIKVIK
Lys1
-11.3
1
uM
5z-7-oxozeaenol BCWM.1 LATS1
ALYATKTLR
Lys1
11.3
1
uM
5z-7-oxozeaenol MWCL.1 MAP2K4
DIKPSNILLDR
Lys2
-11.4
1
uM
5z-7-oxozeaenol BCWM.1 MASTL
LYAVKVVK
Lys1
11.4
1
uM
5z-7-oxozeaenol BCWM.1 PCTAIRE2,PCTAIRE3
SKLTENLVALKEIR
Lys1
-11.5
1
uM
5z-7-oxozeaenol BCWM.1 MARK3
EVAIKIIDKTQLNPTSLQK
Lys1
11.5
1
uM
5z-7-oxozeaenol MWCL.1 MAP3K5
DIKGDNVLINTYSGVLK
Lys2
11.5
1
uM
5z-7-oxozeaenol MWCL.1 RSK3_domain1
DLKPENILLDEEGHIKITDFGLSK
Lys2
11.6
1
uM
5z-7-oxozeaenol MWCL.1 PHKg1
DLKPENILLDDNMNIK
Lys2
-11.8
1
uM
5z-7-oxozeaenol BCWM.1 PKD2
DVAVKVIDK
Lys1
11.8
1
uM
5z-7-oxozeaenol MWCL.1 GSK3A
DIKPQNLLVDPDTAVLK
Lys2
-11.9
1
uM
5z-7-oxozeaenol MWCL.1 NEK1
DIKSQNIFLTK
Lys2
-11.9
1
uM
5z-7-oxozeaenol BCWM.1 CK1d,CK1e
DVKPDNFLMGLGKK
Lys2
11.9
1
uM
5z-7-oxozeaenol MWCL.1 PKD2
DVAVKVIDK
Lys1
11.9
1
uM
5z-7-oxozeaenol MWCL.1 SRPK1
IIHTDIKPENILLSVNEQYIR
Lys2
-1.2
1
uM
5z-7-oxozeaenol BCWM.1 PLK1
CFEISDADTKEVFAGKIVPK
Lys1
1.2
1
uM
5z-7-oxozeaenol MWCL.1 CDK6
DLKPQNILVTSSGQIK
Lys2
1.2
1
uM