5z-7-oxozeaenol KiNativ -- single dose experiment - Dataset (ID:20255)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
5z-7-oxozeaenol | MWCL.1 | MK01 | DLKPSNLLLNTTCDLK | Lys2 | 1.1 | 1 | uM |
5z-7-oxozeaenol | MWCL.1 | MST1 | ETGQIVAIKQVPVESDLQEIIK | Lys1 | -11.0 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | LATS2 | DIKPDNILIDLDGHIK | Lys2 | -11.0 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | GCN2_domain2 | DLKPVNIFLDSDDHVK | Lys2 | 11.0 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | CAMK1D | LFAVKCIPK | Lys1 | 11.1 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | RIPK2 | VQVAVKHLHIHTPLLDSER | Lys1 | 11.1 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | TYK2(Kin.Dom.2) | IGDFGLAKAVPEGHEYYR | Activation Loop | 11.1 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | SNRK | DLKPENVVFFEK | Lys2 | -11.3 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | M4K3 | NVNTGELAAIKVIK | Lys1 | -11.3 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | LATS1 | ALYATKTLR | Lys1 | 11.3 | 1 | uM |
5z-7-oxozeaenol | MWCL.1 | MAP2K4 | DIKPSNILLDR | Lys2 | -11.4 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | MASTL | LYAVKVVK | Lys1 | 11.4 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | PCTAIRE2,PCTAIRE3 | SKLTENLVALKEIR | Lys1 | -11.5 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | MARK3 | EVAIKIIDKTQLNPTSLQK | Lys1 | 11.5 | 1 | uM |
5z-7-oxozeaenol | MWCL.1 | MAP3K5 | DIKGDNVLINTYSGVLK | Lys2 | 11.5 | 1 | uM |
5z-7-oxozeaenol | MWCL.1 | RSK3_domain1 | DLKPENILLDEEGHIKITDFGLSK | Lys2 | 11.6 | 1 | uM |
5z-7-oxozeaenol | MWCL.1 | PHKg1 | DLKPENILLDDNMNIK | Lys2 | -11.8 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | PKD2 | DVAVKVIDK | Lys1 | 11.8 | 1 | uM |
5z-7-oxozeaenol | MWCL.1 | GSK3A | DIKPQNLLVDPDTAVLK | Lys2 | -11.9 | 1 | uM |
5z-7-oxozeaenol | MWCL.1 | NEK1 | DIKSQNIFLTK | Lys2 | -11.9 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | CK1d,CK1e | DVKPDNFLMGLGKK | Lys2 | 11.9 | 1 | uM |
5z-7-oxozeaenol | MWCL.1 | PKD2 | DVAVKVIDK | Lys1 | 11.9 | 1 | uM |
5z-7-oxozeaenol | MWCL.1 | SRPK1 | IIHTDIKPENILLSVNEQYIR | Lys2 | -1.2 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | PLK1 | CFEISDADTKEVFAGKIVPK | Lys1 | 1.2 | 1 | uM |
5z-7-oxozeaenol | MWCL.1 | CDK6 | DLKPQNILVTSSGQIK | Lys2 | 1.2 | 1 | uM |