5z-7-oxozeaenol KiNativ -- single dose experiment - Dataset (ID:20255)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| 5z-7-oxozeaenol | MWCL.1 | NDR2 | DIKPDNLLLDAK | Lys2 | -3.9 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | MAST1,MAST2 | DLKPDNLLITSMGHIK | Lys2 | 39.2 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | PEK | DLKPSNIFFTMDDVVK | Lys2 | 39.8 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | RIPK3 | DLKPSNVLLDPELHVK | Lys2 | -4.0 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | KCC2D | IPTGQEYAAKIINTKK | Lys1 | 4.0 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | RSKL1_domain1 | VLGVIDKVLLVMDTR | Protein Kinase Domain | 4.0 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | ZC2/TNIK | TGQLAAIKVMDVTGDEEEEIKQEINMLKK | Lys1 | 40.1 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | AurA | FILALKVLFK | Lys1 | -4.1 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | MK01 | DLKPSNLLLNTTCDLK | Lys2 | 4.1 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | MK03 | DLKPSNLLINTTCDLK | Lys2 | 4.1 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | DNAPK | EHPFLVKGGEDLR | ATP | 41.3 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | MAST1,MAST2 | DLKPDNLLITSMGHIK | Lys2 | 41.6 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | CDK5 | DLKPQNLLINR | Lys2 | -4.2 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | MARK3 | EVAIKIIDKTQLNPTSLQK | Lys1 | -4.4 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | PKR | DLKPSNIFLVDTK | Lys2 | -4.4 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | KS6B1 | DLKPENIMLNHQGHVK | Lys2 | -44.1 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | GCN2_domain2 | DLKPVNIFLDSDDHVK | Lys2 | 4.5 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | KSR1,KSR2 | SKNVFYDNGK | Activation Loop | 45.0 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | LRRK2 | DLKPHNVLLFTLYPNAAIIAK | Lys2 | -4.6 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | PI4KA,PI4KAP2 | SGTPMQSAAKAPYLAK | ATP | 46.0 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | M3K2,MAP3K3 | DIKGANILR | Lys2 | -4.7 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | ZC2/TNIK | TGQLAAIKVMDVTGDEEEEIKQEINMLKK | Lys1 | 47.5 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | LOK | DLKAGNVLMTLEGDIR | Lys2 | 47.7 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | FYV1 | GGKSGAAFYATEDDRFILK | ATP | 4.8 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | PHKg2 | ATGHEFAVKIMEVTAER | Lys1 | 4.8 | 1 | uM |