5z-7-oxozeaenol KiNativ -- single dose experiment - Dataset (ID:20255)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| 5z-7-oxozeaenol | BCWM.1 | FAK2 | YIEDEDYYKASVTR | Activation Loop | 27.1 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | CSK | VSDFGLTKEASSTQDTGKLPVK | Activation Loop | -3.5 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | BTK | YVLDDEYTSSVGSKFPVR | Activation Loop | -1.6 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | CSK | VSDFGLTKEASSTQDTGKLPVK | Activation Loop | 3.6 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | BTK | YVLDDEYTSSVGSKFPVR | Activation Loop | -2.2 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | ABL,ARG | LMTGDTYTAHAGAKFPIK | Activation Loop | 25.5 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | FGR | LIKDDEYNPCQGSKFPIK | Activation Loop | 16.3 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | FYN,SRC,YES | QGAKFPIKWTAPEAALYGR | Activation Loop | 18.4 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | EPHB1 | YLQDDTSDPTYTSSLGGKIPVR | Activation Loop | 7.7 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | EPHB2 | FLEDDTSDPTYTSALGGKIPIR | Activation Loop | 8.8 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | KSR1,KSR2 | SKNVFYDNGK | Activation Loop | 59.5 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | JAK3 domain2 | IADFGLAKLLPLDKDYYVVR | Activation Loop | 21.6 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | KSR1 | SKNVFYDNGKVVITDFGLFGISGVVR | Activation Loop | 51.6 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | LCK | EGAKFPIKWTAPEAINYGTFTIK | Activation Loop | 15.6 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | STLK5 | YSVKVLPWLSPEVLQQNLQGYDAK | Activation Loop | 2.7 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | DGKA | IDPVPNTHPLLVFVNPKSGGK | ATP | -5.1 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | PI42C | TLVIKEVSSEDIADMHSNLSNYHQYIVK | ATP | 22.2 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | ATR | FYIMMCKPK | ATP | 28.5 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | PAN3 | VMDPTKILITGK | ATP | 5.9 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | ATR | FYIMMCKPK | ATP | 28.8 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | PI4KA,PI4KAP2 | SGTPMQSAAKAPYLAK | ATP | 32.3 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | DGKA | IDPVPNTHPLLVFVNPKSGGK | ATP | -18.8 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | DNAPK | EHPFLVKGGEDLR | ATP | 41.3 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | SMG1 | DTVTIHSVGGTITILPTKTKPK | ATP | 15.7 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | PIP4K2A | AKELPTLKDNDFINEGQK | ATP | 14.2 | 1 | uM |