5z-7-oxozeaenol KiNativ -- single dose experiment - Dataset (ID:20255)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
5z-7-oxozeaenol BCWM.1 NDR2
DIKPDNLLLDAK
Lys2
2.8
1
uM
5z-7-oxozeaenol BCWM.1 NEK1
DIKSQNIFLTK
Lys2
9.4
1
uM
5z-7-oxozeaenol BCWM.1 NEK2
DLKPANVFLDGK
Lys2
15.9
1
uM
5z-7-oxozeaenol BCWM.1 NEK4
DLKTQNVFLTR
Lys2
8.1
1
uM
5z-7-oxozeaenol BCWM.1 NEK6,NEK7
DIKPANVFITATGVVK
Lys2
7.1
1
uM
5z-7-oxozeaenol BCWM.1 NEK8
DLKTQNILLDK
Lys2
-1.7
1
uM
5z-7-oxozeaenol BCWM.1 NEK9
DIKTLNIFLTK
Lys2
15.6
1
uM
5z-7-oxozeaenol BCWM.1 OSR1
DVKAGNILLGEDGSVQIADFGVSAFLATGGDITR
Lys2
9.3
1
uM
5z-7-oxozeaenol BCWM.1 p38a
DLKPSNLAVNEDCELK
Lys2
13.8
1
uM
5z-7-oxozeaenol BCWM.1 p38d,p38g
DLKPGNLAVNEDCELK
Lys2
-0.7
1
uM
5z-7-oxozeaenol BCWM.1 PEK
DLKPSNIFFTMDDVVK
Lys2
17.7
1
uM
5z-7-oxozeaenol BCWM.1 PHKg1
DLKPENILLDDNMNIK
Lys2
-1.8
1
uM
5z-7-oxozeaenol BCWM.1 PITSLRE
DLKTSNLLLSHAGILK
Lys2
2.3
1
uM
5z-7-oxozeaenol BCWM.1 PKR
DLKPSNIFLVDTK
Lys2
7.4
1
uM
5z-7-oxozeaenol BCWM.1 PRP4
CNILHADIKPDNILVNESK
Lys2
1.7
1
uM
5z-7-oxozeaenol BCWM.1 RIPK3
DLKPSNVLLDPELHVK
Lys2
-4.0
1
uM
5z-7-oxozeaenol BCWM.1 ROCK1,ROCK2
DVKPDNMLLDK
Lys2
22.9
1
uM
5z-7-oxozeaenol BCWM.1 RSK1 domain1
DLKPENILLDEEGHIKLTDFGLSKEAIDHEK
Lys2
12.7
1
uM
5z-7-oxozeaenol BCWM.1 RSK2 domain1
DLKPENILLDEEGHIKLTDFGLSKESIDHEK
Lys2
23.5
1
uM
5z-7-oxozeaenol BCWM.1 RSK4 domain1
DLKPENILLDEIGHIK
Lys2
25.6
1
uM
5z-7-oxozeaenol BCWM.1 SLK
DLKAGNILFTLDGDIK
Lys2
-2.3
1
uM
5z-7-oxozeaenol BCWM.1 SNRK
DLKPENVVFFEK
Lys2
-11.3
1
uM
5z-7-oxozeaenol BCWM.1 SRPK1
IIHTDIKPENILLSVNEQYIR
Lys2
-1.0
1
uM
5z-7-oxozeaenol BCWM.1 STK33
DLKLENIMVK
Lys2
3.1
1
uM
5z-7-oxozeaenol BCWM.1 TLK1
YLNEIKPPIIHYDLKPGNILLVDGTACGEIK
Lys2
-2.3
1
uM