5z-7-oxozeaenol KiNativ -- single dose experiment - Dataset (ID:20255)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
5z-7-oxozeaenol | BCWM.1 | NDR2 | DIKPDNLLLDAK | Lys2 | 2.8 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | NEK1 | DIKSQNIFLTK | Lys2 | 9.4 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | NEK2 | DLKPANVFLDGK | Lys2 | 15.9 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | NEK4 | DLKTQNVFLTR | Lys2 | 8.1 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | NEK6,NEK7 | DIKPANVFITATGVVK | Lys2 | 7.1 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | NEK8 | DLKTQNILLDK | Lys2 | -1.7 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | NEK9 | DIKTLNIFLTK | Lys2 | 15.6 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | OSR1 | DVKAGNILLGEDGSVQIADFGVSAFLATGGDITR | Lys2 | 9.3 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | p38a | DLKPSNLAVNEDCELK | Lys2 | 13.8 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | p38d,p38g | DLKPGNLAVNEDCELK | Lys2 | -0.7 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | PEK | DLKPSNIFFTMDDVVK | Lys2 | 17.7 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | PHKg1 | DLKPENILLDDNMNIK | Lys2 | -1.8 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | PITSLRE | DLKTSNLLLSHAGILK | Lys2 | 2.3 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | PKR | DLKPSNIFLVDTK | Lys2 | 7.4 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | PRP4 | CNILHADIKPDNILVNESK | Lys2 | 1.7 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | RIPK3 | DLKPSNVLLDPELHVK | Lys2 | -4.0 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | ROCK1,ROCK2 | DVKPDNMLLDK | Lys2 | 22.9 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | RSK1 domain1 | DLKPENILLDEEGHIKLTDFGLSKEAIDHEK | Lys2 | 12.7 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | RSK2 domain1 | DLKPENILLDEEGHIKLTDFGLSKESIDHEK | Lys2 | 23.5 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | RSK4 domain1 | DLKPENILLDEIGHIK | Lys2 | 25.6 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | SLK | DLKAGNILFTLDGDIK | Lys2 | -2.3 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | SNRK | DLKPENVVFFEK | Lys2 | -11.3 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | SRPK1 | IIHTDIKPENILLSVNEQYIR | Lys2 | -1.0 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | STK33 | DLKLENIMVK | Lys2 | 3.1 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | TLK1 | YLNEIKPPIIHYDLKPGNILLVDGTACGEIK | Lys2 | -2.3 | 1 | uM |