5z-7-oxozeaenol KiNativ -- single dose experiment - Dataset (ID:20255)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| 5z-7-oxozeaenol | MWCL.1 | JAK3 domain2 | IADFGLAKLLPLDKDYYVVR | Activation Loop | 33.9 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | JNK1,JNK2,JNK3 | DLKPSNIVVK | Lys2 | -2.3 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | KHS1 | NVHTGELAAVKIIK | Lys1 | -15.8 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | KSR1 | SKNVFYDNGKVVITDFGLFGISGVVR | Activation Loop | 61.6 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | KSR1,KSR2 | SKNVFYDNGK | Activation Loop | 45.0 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | LATS1 | ALYATKTLR | Lys1 | -5.3 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | LATS2 | DIKPDNILIDLDGHIK | Lys2 | 1 | uM | |
| 5z-7-oxozeaenol | MWCL.1 | LCK | EGAKFPIKWTAPEAINYGTFTIK | Activation Loop | 33.1 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | LKB1 | DIKPGNLLLTTGGTLK | Lys2 | 0.0 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | LOK | DLKAGNVLMTLEGDIR | Lys2 | 47.7 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | LRRK2 | DLKPHNVLLFTLYPNAAIIAK | Lys2 | -4.6 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | LYN | VAVKTLKPGTMSVQAFLEEANLMK | Lys1 | 1 | uM | |
| 5z-7-oxozeaenol | MWCL.1 | MAP2K1 | IMHRDVKPSNILVNSR | Lys2 | 91.2 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | MAP2K1,MAP2K2 | DVKPSNILVNSR | Lys2 | 93.7 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | MAP2K3 | DVKPSNVLINK | Lys2 | 35.6 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | MAP2K4 | DIKPSNILLDR | Lys2 | -11.4 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | MAP2K5 | DVKPSNMLVNTR | Lys2 | 75.1 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | MAP2K6 | DVKPSNVLINALGQVK | Lys2 | 73.9 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | MAP3K1 | DVKGANLLIDSTGQR | Lys2 | 25.6 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | MAP3K3 | ELASKQVQFDPDSPETSKEVSALECEIQLLK | Lys1 | -6.2 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | MAP3K4 | DIKGANIFLTSSGLIK | Lys2 | 8.3 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | MAP3K5 | DIKGDNVLINTYSGVLK | Lys2 | 11.5 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | M3K6 | DIKGDNVLINTFSGLLK | Lys2 | -9.5 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | MARK2,MARK3 | DLKAENLLLDADMNIK | Lys2 | 29.7 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | MARK3 | EVAIKIIDKTQLNPTSLQK | Lys1 | -4.4 | 1 | uM |