PF-3758309 KiNativ -- single dose experiment - Dataset (ID:20254)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
PF-3758309 | THP-1 | IKKE | SGELVAVKVFNTTSYLRPR | Lys1 | 87.7 | 1 | uM |
PF-3758309 | THP-1 | PCTAIRE2,PCTAIRE3 | SKLTENLVALKEIR | Lys1 | 73.1 | 1 | uM |
PF-3758309 | THP-1 | NEK3 | SKNIFLTQNGK | Activation Loop | -1.7 | 1 | uM |
PF-3758309 | THP-1 | NEK9 | TEDDSLVVWKEVDLTR | Lys1 | 21.4 | 1 | uM |
PF-3758309 | THP-1 | PI42C | TLVIKEVSSEDIADMHSNLSNYHQYIVK | ATP | -20.7 | 1 | uM |
PF-3758309 | THP-1 | CaMK2g | TSTQEYAAKIINTK | Lys1 | 89.3 | 1 | uM |
PF-3758309 | THP-1 | FER | TSVAVKTCKEDLPQELK | Lys1 | 73.7 | 1 | uM |
PF-3758309 | THP-1 | SYK | TVAVKILK | Lys1 | 6.7 | 1 | uM |
PF-3758309 | THP-1 | ACK | TVSVAVKCLKPDVLSQPEAMDDFIR | Lys1 | 1.9 | 1 | uM |
PF-3758309 | THP-1 | SIK3 | VAIKIIDKTQLDEENLKK | Lys1 | 25.0 | 1 | uM |
PF-3758309 | THP-1 | CHK2 | VAIKIISK | Lys1 | 91.1 | 1 | uM |
PF-3758309 | THP-1 | AMPKa1,AMPKa2 | VAVKILNR | Lys1 | 97.6 | 1 | uM |
PF-3758309 | THP-1 | INSR | VAVKTVNESASLR | Lys1 | 9.1 | 1 | uM |
PF-3758309 | THP-1 | PIK3CB | VFGEDSVGVIFKNGDDLR | ATP | 7.1 | 1 | uM |
PF-3758309 | THP-1 | PKN1 | VLLSEFRPSGELFAIKALK | Lys1 | 68.6 | 1 | uM |
PF-3758309 | THP-1 | PIK3CD | VNWLAHNVSKDNRQ | ATP | -0.4 | 1 | uM |
PF-3758309 | THP-1 | CSK | VSDFGLTKEASSTQDTGKLPVK | Activation Loop | 12.7 | 1 | uM |
PF-3758309 | THP-1 | IKKB | WHNQETGEQIAIKQCR | Lys1 | 2.5 | 1 | uM |
PF-3758309 | THP-1 | MLTK | WISQDKEVAVKK | Lys1 | -6.3 | 1 | uM |
PF-3758309 | THP-1 | ILK | WQGNDIVVKVLK | Lys1 | -3.6 | 1 | uM |
PF-3758309 | THP-1 | FAK2 | YIEDEDYYKASVTR | Activation Loop | 63.9 | 1 | uM |
PF-3758309 | THP-1 | eEF2K | YIKYNSNSGFVR | ATP | -2.2 | 1 | uM |
PF-3758309 | THP-1 | TLK2 | YVAVKIHQLNK | Lys1 | 64.3 | 1 | uM |
PF-3758309 | THP-1 | BTK | YVLDDEYTSSVGSKFPVR | Activation Loop | -2.7 | 1 | uM |