PF-3758309 KiNativ -- single dose experiment - Dataset (ID:20254)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| PF-3758309 | THP-1 | CDK20 | DLKPANLLISASGQLK | Lys2 | 7.1 | 1 | uM |
| PF-3758309 | THP-1 | RSK1,RSK2,RSK3_domain1 | DLKPENILLDEEGHIK | Lys2 | 90.6 | 1 | uM |
| PF-3758309 | THP-1 | CDK4 | DLKPENILVTSGGTVK | Lys2 | -8.8 | 1 | uM |
| PF-3758309 | THP-1 | KS6B1 | DLKPENIMLNHQGHVK | Lys2 | -8.0 | 1 | uM |
| PF-3758309 | THP-1 | CaMK2a,CaMK2b,CaMK2d,CaMK2g | DLKPENLLLASK | Lys2 | 79.9 | 1 | uM |
| PF-3758309 | THP-1 | AMPKa1,AMPKa2 | DLKPENVLLDAHMNAK | Lys2 | 96.4 | 1 | uM |
| PF-3758309 | THP-1 | CHK2 | DLKPENVLLSSQEEDCLIK | Lys2 | 81.8 | 1 | uM |
| PF-3758309 | THP-1 | SNRK | DLKPENVVFFEK | Lys2 | -7.9 | 1 | uM |
| PF-3758309 | THP-1 | p38d,p38g | DLKPGNLAVNEDCELK | Lys2 | 5.2 | 1 | uM |
| PF-3758309 | THP-1 | CDK7 | DLKPNNLLLDENGVLK | Lys2 | 96.5 | 1 | uM |
| PF-3758309 | THP-1 | ULK1 | DLKPQNILLSNPAGR | Lys2 | -9.5 | 1 | uM |
| PF-3758309 | THP-1 | CDK6 | DLKPQNILVTSSGQIK | Lys2 | -6.4 | 1 | uM |
| PF-3758309 | THP-1 | CDC2 | DLKPQNLLIDDKGTIK | Lys2 | -0.9 | 1 | uM |
| PF-3758309 | THP-1 | PCTAIRE2 | DLKPQNLLINEK | Lys2 | 70.0 | 1 | uM |
| PF-3758309 | THP-1 | CDK16 | DLKPQNLLINER | Lys2 | 63.7 | 1 | uM |
| PF-3758309 | THP-1 | CDK5 | DLKPQNLLINR | Lys2 | -31.5 | 1 | uM |
| PF-3758309 | THP-1 | CDK2 | DLKPQNLLINTEGAIK | Lys2 | 2.8 | 1 | uM |
| PF-3758309 | THP-1 | PKR | DLKPSNIFLVDTK | Lys2 | 2.3 | 1 | uM |
| PF-3758309 | THP-1 | RSK2_domain2 | DLKPSNILYVDESGNPESIR | Lys2 | -6.9 | 1 | uM |
| PF-3758309 | THP-1 | JNK1,JNK2,JNK3 | DLKPSNIVVK | Lys2 | 1.0 | 1 | uM |
| PF-3758309 | THP-1 | p38a | DLKPSNLAVNEDCELK | Lys2 | 1.1 | 1 | uM |
| PF-3758309 | THP-1 | MK03 | DLKPSNLLINTTCDLK | Lys2 | 56.5 | 1 | uM |
| PF-3758309 | THP-1 | MK01 | DLKPSNLLLNTTCDLK | Lys2 | 55.4 | 1 | uM |
| PF-3758309 | THP-1 | RIPK3 | DLKPSNVLLDPELHVK | Lys2 | -14.0 | 1 | uM |
| PF-3758309 | THP-1 | BRAF | DLKSNNIFLHEDLTVK | Lys2 | -5.4 | 1 | uM |