PF-3758309 KiNativ -- single dose experiment - Dataset (ID:20254)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| PF-3758309 | THP-1 | SLK | DLKAGNILFTLDGDIK | Lys2 | 17.6 | 1 | uM |
| PF-3758309 | THP-1 | CDK5 | DLKPQNLLINR | Lys2 | -31.5 | 1 | uM |
| PF-3758309 | THP-1 | IRAK1 | AIQFLHQDSPSLIHGDIKSSNVLLDER | Lys2 | 8.6 | 1 | uM |
| PF-3758309 | THP-1 | IRAK4 | DIKSANILLDEAFTAK | Lys2 | 4.0 | 1 | uM |
| PF-3758309 | THP-1 | JNK1,JNK2,JNK3 | DLKPSNIVVK | Lys2 | 1.0 | 1 | uM |
| PF-3758309 | THP-1 | CDK4 | DLKPENILVTSGGTVK | Lys2 | -8.8 | 1 | uM |
| PF-3758309 | THP-1 | CDK2 | DLKPQNLLINTEGAIK | Lys2 | 2.8 | 1 | uM |
| PF-3758309 | THP-1 | LKB1 | DIKPGNLLLTTGGTLK | Lys2 | 84.9 | 1 | uM |
| PF-3758309 | THP-1 | CDK11,CDK8 | DLKPANILVMGEGPER | Lys2 | -29.4 | 1 | uM |
| PF-3758309 | THP-1 | MAP2K1,MAP2K2 | DVKPSNILVNSR | Lys2 | -6.6 | 1 | uM |
| PF-3758309 | THP-1 | MAP2K3 | DVKPSNVLINK | Lys2 | -7.5 | 1 | uM |
| PF-3758309 | THP-1 | CDC2 | DLKPQNLLIDDKGTIK | Lys2 | -0.9 | 1 | uM |
| PF-3758309 | THP-1 | MAP2K5 | DVKPSNMLVNTR | Lys2 | -18.2 | 1 | uM |
| PF-3758309 | THP-1 | SNRK | DLKPENVVFFEK | Lys2 | -7.9 | 1 | uM |
| PF-3758309 | THP-1 | MAP2K6 | DVKPSNVLINALGQVK | Lys2 | 21.2 | 1 | uM |
| PF-3758309 | THP-1 | MP2K7 | DVKPSNILLDER | Lys2 | 14.7 | 1 | uM |
| PF-3758309 | THP-1 | MAP3K1 | DVKGANLLIDSTGQR | Lys2 | -9.4 | 1 | uM |
| PF-3758309 | THP-1 | M3K2,MAP3K3 | DIKGANILR | Lys2 | 10.7 | 1 | uM |
| PF-3758309 | THP-1 | ZC1/HGK,ZC2/TNIK,ZC3/MINK | DIKGQNVLLTENAEVK | Lys2 | 8.4 | 1 | uM |
| PF-3758309 | THP-1 | PKR | DLKPSNIFLVDTK | Lys2 | 2.3 | 1 | uM |
| PF-3758309 | THP-1 | Wnk1,Wnk2,Wnk3 | DLKCDNIFITGPTGSVK | Lys2 | 0.9 | 1 | uM |
| PF-3758309 | THP-1 | CDK7 | DLKPNNLLLDENGVLK | Lys2 | 96.5 | 1 | uM |
| PF-3758309 | THP-1 | MLK3 | DLKSNNILLLQPIESDDMEHK | Lys2 | 45.0 | 1 | uM |
| PF-3758309 | THP-1 | MK14 | QELNKTIWEVPER | Protein Kinase Domain | 7.4 | 1 | uM |