WZ3105 KiNativ -- single dose experiment - Dataset (ID:20253)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| WZ3105 | THP-1 | PRPK | FLSGLELVKQGAEAR | ATP Loop | 7.1 | 1 | uM |
| WZ3105 | THP-1 | FAK2 | YIEDEDYYKASVTR | Activation Loop | 55.8 | 1 | uM |
| WZ3105 | THP-1 | SIK3 | VAIKIIDKTQLDEENLKK | Lys1 | 7.4 | 1 | uM |
| WZ3105 | THP-1 | RIPK3 | DLKPSNVLLDPELHVK | Lys2 | -28.5 | 1 | uM |
| WZ3105 | THP-1 | RSK1,RSK2,RSK3_domain1 | DLKPENILLDEEGHIK | Lys2 | 50.1 | 1 | uM |
| WZ3105 | THP-1 | RSK1 (Domain 2) | ATNMEYAVKVIDK | Lys1 | 5.2 | 1 | uM |
| WZ3105 | THP-1 | RSK2_domain2 | DLKPSNILYVDESGNPESIR | Lys2 | -12.3 | 1 | uM |
| WZ3105 | THP-1 | SGK3 | FYAVKVLQK | Lys1 | -23.6 | 1 | uM |
| WZ3105 | THP-1 | SLK | DLKAGNILFTLDGDIK | Lys2 | 18.7 | 1 | uM |
| WZ3105 | THP-1 | SNRK | DLKPENVVFFEK | Lys2 | -6.1 | 1 | uM |
| WZ3105 | THP-1 | SRPK1/2 | FVAMKVVK | Lys1 | 24.0 | 1 | uM |
| WZ3105 | THP-1 | STLK6 | HTPTGTLVTIKITNLENCNEER | Lys1 | -1.3 | 1 | uM |
| WZ3105 | THP-1 | SYK | TVAVKILK | Lys1 | -9.9 | 1 | uM |
| WZ3105 | THP-1 | TLK2 | YVAVKIHQLNK | Lys1 | -9.6 | 1 | uM |
| WZ3105 | THP-1 | ULK1 | DLKPQNILLSNPAGR | Lys2 | -11.4 | 1 | uM |
| WZ3105 | THP-1 | ULK3 | EVVAIKCVAK | Lys1 | -5.3 | 1 | uM |
| WZ3105 | THP-1 | Wnk1,Wnk2,Wnk3 | DLKCDNIFITGPTGSVK | Lys2 | -10.2 | 1 | uM |
| WZ3105 | THP-1 | Wnk1,Wnk2,Wnk4 | IGDLGLATLKR | Activation Loop | -9.3 | 1 | uM |
| WZ3105 | THP-1 | MLTK | WISQDKEVAVKK | Lys1 | -9.2 | 1 | uM |
| WZ3105 | THP-1 | ZC1/HGK,ZC2/TNIK,ZC3/MINK | DIKGQNVLLTENAEVK | Lys2 | 18.3 | 1 | uM |
| WZ3105 | THP-1 | M4K3 | NVNTGELAAIKVIK | Lys1 | 28.3 | 1 | uM |
| WZ3105 | THP-1 | MAP3K5,MAP3K6,MAP3K7 | IAIKEIPERDSR | Lys1 | -13.7 | 1 | uM |
| WZ3105 | THP-1 | MARK3 | EVAIKIIDKTQLNPTSLQK | Lys1 | 3.6 | 1 | uM |
| WZ3105 | THP-1 | PIP4K2A | AKELPTLKDNDFINEGQK | ATP | -2.5 | 1 | uM |