Phosphorylation state and protein levels measured in BRAF(V600E/D) melanoma cell lines monitored by imaging - Dataset (ID:20219)
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Small Molecule | Cell Line | 2nd Drug | Drug Concentration | Conc Unit | Time Point | Time Point Unit | Image | Measured Protein (Alexa Fluor 488) | Measured Protein Value (488) | Measured Protein (Alexa Fluor 568) | Measured Protein Value (568) | Measured Protein (Alexa Fluor 647) | Measured Protein Value (647) | Replicate | Plate Name | Plate Well |
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Vemurafenib | COLO 858 | JNK-IN-8 | 0.0512 | uM | 24 | hr | p-Histone H3(S10) | 239.08 | p-Rb(S807/S811) | 140.42 | p-S6(S235/S236 | 380.85 | 2 | Colo858-signal2 | G7 | |
Vemurafenib | COLO 858 | JNK-IN-8 | 0.0033 | uM | 24 | hr | Ki-67 | 2257.40 | p-Rb(S807/S811) | 152.83 | p-cJun(S73) | 28.15 | 1 | Colo858-signal3 | F10 | |
Vemurafenib | COLO 858 | JNK-IN-8 | 0.0000 | uM | 24 | hr | Ki-67 | 2257.00 | p-Rb(S807/S811) | 151.09 | p-cJun(S73) | 29.94 | 1 | Colo858-signal3 | F11 | |
Vemurafenib | COLO 858 | JNK-IN-8 | 2.0000 | uM | 24 | hr | Ki-67 | 1130.80 | p-Rb(S807/S811) | 51.60 | p-cJun(S73) | 14.98 | 1 | Colo858-signal3 | F3 | |
Vemurafenib | COLO 858 | JNK-IN-8 | 0.8000 | uM | 24 | hr | Ki-67 | 807.26 | p-Rb(S807/S811) | 48.49 | p-cJun(S73) | 14.54 | 1 | Colo858-signal3 | F4 | |
Vemurafenib | COLO 858 | JNK-IN-8 | 0.0033 | uM | 24 | hr | p27 Kip1 | 421.06 | p-Rb(S807/S811) | 154.67 | p-ERK(T202/Y204) | 537.34 | 2 | Colo858-signal1 | G10 | |
Vemurafenib | COLO 858 | JNK-IN-8 | 0.0000 | uM | 24 | hr | p27 Kip1 | 447.88 | p-Rb(S807/S811) | 161.30 | p-ERK(T202/Y204) | 568.39 | 2 | Colo858-signal1 | G11 | |
Vemurafenib | COLO 858 | JNK-IN-8 | 2.0000 | uM | 24 | hr | p27 Kip1 | 1676.60 | p-Rb(S807/S811) | 60.57 | p-ERK(T202/Y204) | 20.44 | 2 | Colo858-signal1 | G3 | |
Vemurafenib | COLO 858 | JNK-IN-8 | 0.8000 | uM | 24 | hr | p27 Kip1 | 1044.90 | p-Rb(S807/S811) | 48.21 | p-ERK(T202/Y204) | 22.38 | 2 | Colo858-signal1 | G4 | |
Vemurafenib | COLO 858 | JNK-IN-8 | 0.0512 | uM | 24 | hr | p27 Kip1 | 511.00 | p-Rb(S807/S811) | 125.23 | p-ERK(T202/Y204) | 254.95 | 2 | Colo858-signal1 | G7 | |
Vemurafenib | COLO 858 | JNK-IN-8 | 0.0205 | uM | 24 | hr | p27 Kip1 | 458.83 | p-Rb(S807/S811) | 152.02 | p-ERK(T202/Y204) | 459.90 | 2 | Colo858-signal1 | G8 | |
Vemurafenib | COLO 858 | JNK-IN-8 | 0.0033 | uM | 24 | hr | p-Histone H3(S10) | 288.89 | p-Rb(S807/S811) | 152.75 | p-S6(S235/S236 | 379.48 | 1 | Colo858-signal2 | F10 | |
Vemurafenib | COLO 858 | JNK-IN-8 | 0.0082 | uM | 24 | hr | p27 Kip1 | 461.45 | p-Rb(S807/S811) | 160.46 | p-ERK(T202/Y204) | 599.65 | 1 | Colo858-signal1 | F9 | |
Vemurafenib | COLO 858 | JNK-IN-8 | 0.8000 | uM | 24 | hr | p-Histone H3(S10) | 168.97 | p-Rb(S807/S811) | 57.67 | p-S6(S235/S236 | 47.25 | 1 | Colo858-signal2 | F4 | |
Vemurafenib | COLO 858 | JNK-IN-8 | 0.0033 | uM | 24 | hr | p27 Kip1 | 459.60 | p-Rb(S807/S811) | 160.13 | p-ERK(T202/Y204) | 573.25 | 1 | Colo858-signal1 | F10 | |
Vemurafenib | COLO 858 | JNK-IN-8 | 0.0000 | uM | 24 | hr | p27 Kip1 | 453.65 | p-Rb(S807/S811) | 157.18 | p-ERK(T202/Y204) | 608.40 | 1 | Colo858-signal1 | F11 | |
Vemurafenib | COLO 858 | JNK-IN-8 | 5.0000 | uM | 24 | hr | p27 Kip1 | 1646.10 | p-Rb(S807/S811) | 108.76 | p-ERK(T202/Y204) | 29.73 | 1 | Colo858-signal1 | F2 | |
Vemurafenib | COLO 858 | JNK-IN-8 | 2.0000 | uM | 24 | hr | p27 Kip1 | 1532.60 | p-Rb(S807/S811) | 62.03 | p-ERK(T202/Y204) | 22.35 | 1 | Colo858-signal1 | F3 | |
Vemurafenib | COLO 858 | JNK-IN-8 | 0.8000 | uM | 24 | hr | p27 Kip1 | 1176.20 | p-Rb(S807/S811) | 47.97 | p-ERK(T202/Y204) | 25.00 | 1 | Colo858-signal1 | F4 | |
Vemurafenib | COLO 858 | JNK-IN-8 | 0.3200 | uM | 24 | hr | p27 Kip1 | 1024.70 | p-Rb(S807/S811) | 48.87 | p-ERK(T202/Y204) | 30.22 | 1 | Colo858-signal1 | F5 | |
Vemurafenib | COLO 858 | JNK-IN-8 | 0.1280 | uM | 24 | hr | p27 Kip1 | 738.58 | p-Rb(S807/S811) | 81.58 | p-ERK(T202/Y204) | 80.67 | 1 | Colo858-signal1 | F6 | |
Vemurafenib | COLO 858 | JNK-IN-8 | 0.0512 | uM | 24 | hr | p27 Kip1 | 537.76 | p-Rb(S807/S811) | 125.84 | p-ERK(T202/Y204) | 268.22 | 1 | Colo858-signal1 | F7 | |
Vemurafenib | COLO 858 | JNK-IN-8 | 0.0205 | uM | 24 | hr | p27 Kip1 | 462.46 | p-Rb(S807/S811) | 154.40 | p-ERK(T202/Y204) | 499.08 | 1 | Colo858-signal1 | F8 | |
Vemurafenib | COLO 858 | JNK-IN-8 | 0.0082 | uM | 24 | hr | Ki-67 | 2177.30 | p-Rb(S807/S811) | 151.57 | p-cJun(S73) | 28.39 | 1 | Colo858-signal3 | F9 | |
Vemurafenib | COLO 858 | JNK-IN-8 | 0.0205 | uM | 24 | hr | Ki-67 | 2146.20 | p-Rb(S807/S811) | 150.60 | p-cJun(S73) | 28.79 | 1 | Colo858-signal3 | F8 |