Phosphorylation state and protein levels measured in BRAF(V600E/D) melanoma cell lines monitored by imaging - Dataset (ID:20219)
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Small Molecule | Cell Line | 2nd Drug | Drug Concentration | Conc Unit | Time Point | Time Point Unit | Image | Measured Protein (Alexa Fluor 488) | Measured Protein Value (488) | Measured Protein (Alexa Fluor 568) | Measured Protein Value (568) | Measured Protein (Alexa Fluor 647) | Measured Protein Value (647) | Replicate | Plate Name | Plate Well |
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Vemurafenib | WM-115 | JNK-IN-8 | 0.8000 | uM | 24 | hr | Ki-67 | 682.82 | p-Rb(S807/S811) | 40.64 | p-cJun(S73) | 20.31 | 2 | WM115-signal3 | G4 | |
Vemurafenib | COLO 858 | 0.8000 | uM | 24 | hr | Ki-67 | 680.51 | p-Rb(S807/S811) | 40.34 | p-cJun(S73) | 71.07 | 2 | Colo858-signal3 | C4 | ||
Vemurafenib | WM-115 | JNK-IN-8 | 0.8000 | uM | 24 | hr | p-Histone H3(S10) | 201.42 | p-Rb(S807/S811) | 39.76 | p-S6(S235/S236 | 56.51 | 1 | WM115-signal2 | F4 | |
Vemurafenib | WM-115 | 0.8000 | uM | 24 | hr | Ki-67 | 663.63 | p-Rb(S807/S811) | 39.63 | p-cJun(S73) | 79.94 | 1 | WM115-signal3 | B4 | ||
Vemurafenib | WM-115 | JNK-IN-8 | 0.8000 | uM | 24 | hr | p27 Kip1 | 302.92 | p-Rb(S807/S811) | 39.51 | p-ERK(T202/Y204) | 28.13 | 2 | WM115-signal1 | G4 | |
Vemurafenib | WM-115 | 0.8000 | uM | 24 | hr | p-Histone H3(S10) | 179.29 | p-Rb(S807/S811) | 38.89 | p-S6(S235/S236 | 65.75 | 2 | WM115-signal2 | C4 | ||
Vemurafenib | WM-115 | JNK-IN-8 | 0.8000 | uM | 24 | hr | p-Histone H3(S10) | 182.61 | p-Rb(S807/S811) | 38.78 | p-S6(S235/S236 | 51.74 | 2 | WM115-signal2 | G4 | |
Vemurafenib | WM-115 | 0.8000 | uM | 24 | hr | p27 Kip1 | 301.62 | p-Rb(S807/S811) | 38.59 | p-ERK(T202/Y204) | 24.54 | 2 | WM115-signal1 | C4 | ||
Vemurafenib | WM-115 | 0.8000 | uM | 24 | hr | p27 Kip1 | 304.70 | p-Rb(S807/S811) | 38.57 | p-ERK(T202/Y204) | 23.27 | 1 | WM115-signal1 | B4 | ||
Vemurafenib | WM-115 | 0.8000 | uM | 24 | hr | Ki-67 | 666.78 | p-Rb(S807/S811) | 38.55 | p-cJun(S73) | 82.82 | 2 | WM115-signal3 | C4 | ||
Vemurafenib | WM-115 | 0.3200 | uM | 24 | hr | Ki-67 | 721.37 | p-Rb(S807/S811) | 38.52 | p-cJun(S73) | 78.48 | 1 | WM115-signal3 | B5 | ||
Vemurafenib | WM-115 | 0.3200 | uM | 24 | hr | p-Histone H3(S10) | 180.39 | p-Rb(S807/S811) | 38.47 | p-S6(S235/S236 | 77.58 | 1 | WM115-signal2 | B5 | ||
Vemurafenib | WM-115 | 0.3200 | uM | 24 | hr | p27 Kip1 | 257.65 | p-Rb(S807/S811) | 38.40 | p-ERK(T202/Y204) | 44.96 | 2 | WM115-signal1 | C5 | ||
Vemurafenib | WM-115 | 0.8000 | uM | 24 | hr | p-Histone H3(S10) | 190.48 | p-Rb(S807/S811) | 38.37 | p-S6(S235/S236 | 66.01 | 1 | WM115-signal2 | B4 | ||
Vemurafenib | WM-115 | 0.3200 | uM | 24 | hr | p27 Kip1 | 263.18 | p-Rb(S807/S811) | 37.97 | p-ERK(T202/Y204) | 43.14 | 1 | WM115-signal1 | B5 | ||
Vemurafenib | WM-115 | JNK-IN-8 | 0.3200 | uM | 24 | hr | p-Histone H3(S10) | 173.97 | p-Rb(S807/S811) | 36.66 | p-S6(S235/S236 | 72.75 | 2 | WM115-signal2 | G5 | |
Vemurafenib | WM-115 | 0.3200 | uM | 24 | hr | p-Histone H3(S10) | 148.64 | p-Rb(S807/S811) | 35.95 | p-S6(S235/S236 | 64.00 | 2 | WM115-signal2 | C5 | ||
Vemurafenib | WM-115 | 0.3200 | uM | 24 | hr | Ki-67 | 587.55 | p-Rb(S807/S811) | 26.27 | p-cJun(S73) | 71.93 | 2 | WM115-signal3 | C5 | ||
Vemurafenib | WM-115 | JNK-IN-8 | 0.0205 | uM | 24 | hr | p-Histone H3(S10) | p-Rb(S807/S811) | p-S6(S235/S236 | 1 | WM115-signal2 | F8 | ||||
Vemurafenib | WM-115 | JNK-IN-8 | 0.0082 | uM | 24 | hr | p-Histone H3(S10) | p-Rb(S807/S811) | p-S6(S235/S236 | 1 | WM115-signal2 | F9 |