Viability and apoptosis in BRAF(V600E/D) melanoma cell lines monitored by imaging - Dataset (ID:20217)
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Small Molecule | Cell Line | Drug Concentration | Conc Unit | Time Point | Time Point Unit | Total Number of Cells (Nuclei) | Number of Apoptotic Cells | Relative Viability | Mean Relative Viability | Apoptosis Fraction | Mean Apoptosis Fraction | Replicate |
---|---|---|---|---|---|---|---|---|---|---|---|---|
AZ-628 | C32 | 3.1600 | uM | 72 | hr | 1133 | 1071 | 0.0271 | 0.0269 | 0.9453 | 0.9414 | 4 |
AZ-628 | C32 | 3.1600 | uM | 72 | hr | 1046 | 997 | 0.0214 | 0.0269 | 0.9532 | 0.9414 | 1 |
AZ-628 | C32 | 3.1600 | uM | 72 | hr | 992 | 934 | 0.0253 | 0.0269 | 0.9415 | 0.9414 | 2 |
AZ-628 | C32 | 3.1600 | uM | 72 | hr | 1035 | 958 | 0.0336 | 0.0269 | 0.9256 | 0.9414 | 3 |
Vemurafenib | C32 | 3.1600 | uM | 72 | hr | 995 | 960 | 0.0153 | 0.0274 | 0.9648 | 0.9276 | 2 |
Vemurafenib | C32 | 3.1600 | uM | 72 | hr | 998 | 921 | 0.0336 | 0.0274 | 0.9229 | 0.9276 | 1 |
Vemurafenib | C32 | 3.1600 | uM | 72 | hr | 775 | 688 | 0.0380 | 0.0274 | 0.8877 | 0.9276 | 3 |
Vemurafenib | C32 | 3.1600 | uM | 72 | hr | 798 | 746 | 0.0227 | 0.0274 | 0.9348 | 0.9276 | 4 |
AZ-628 | C32 | 1.0000 | uM | 72 | hr | 1409 | 1291 | 0.0515 | 0.0591 | 0.9163 | 0.8863 | 2 |
AZ-628 | C32 | 1.0000 | uM | 72 | hr | 1155 | 1032 | 0.0537 | 0.0591 | 0.8935 | 0.8863 | 4 |
AZ-628 | C32 | 1.0000 | uM | 72 | hr | 1138 | 972 | 0.0725 | 0.0591 | 0.8541 | 0.8863 | 3 |
AZ-628 | C32 | 1.0000 | uM | 72 | hr | 1127 | 993 | 0.0585 | 0.0591 | 0.8811 | 0.8863 | 1 |
Selumetinib | C32 | 3.1600 | uM | 72 | hr | 1035 | 878 | 0.0685 | 0.0615 | 0.8483 | 0.8621 | 2 |
Selumetinib | C32 | 3.1600 | uM | 72 | hr | 943 | 840 | 0.0450 | 0.0615 | 0.8908 | 0.8621 | 1 |
Selumetinib | C32 | 3.1600 | uM | 72 | hr | 924 | 822 | 0.0445 | 0.0615 | 0.8896 | 0.8621 | 3 |
Selumetinib | C32 | 3.1600 | uM | 72 | hr | 1114 | 913 | 0.0878 | 0.0615 | 0.8196 | 0.8621 | 4 |
PLX-4720 | C32 | 3.1600 | uM | 72 | hr | 820 | 631 | 0.0825 | 0.0669 | 0.7695 | 0.8134 | 2 |
PLX-4720 | C32 | 3.1600 | uM | 72 | hr | 856 | 729 | 0.0554 | 0.0669 | 0.8516 | 0.8134 | 3 |
PLX-4720 | C32 | 3.1600 | uM | 72 | hr | 873 | 773 | 0.0437 | 0.0669 | 0.8855 | 0.8134 | 1 |
PLX-4720 | C32 | 3.1600 | uM | 72 | hr | 778 | 581 | 0.0860 | 0.0669 | 0.7468 | 0.8134 | 4 |
AZ-628 | C32 | 3.1600 | uM | 48 | hr | 1579 | 1414 | 0.0803 | 0.0749 | 0.8955 | 0.9051 | 3 |
AZ-628 | C32 | 3.1600 | uM | 48 | hr | 1609 | 1466 | 0.0696 | 0.0749 | 0.9111 | 0.9051 | 1 |
AZ-628 | C32 | 3.1600 | uM | 48 | hr | 1553 | 1419 | 0.0652 | 0.0749 | 0.9137 | 0.9051 | 4 |
AZ-628 | C32 | 3.1600 | uM | 48 | hr | 1739 | 1565 | 0.0847 | 0.0749 | 0.8999 | 0.9051 | 2 |
AZ-628 | WM-115 | 3.1600 | uM | 72 | hr | 1146 | 960 | 0.0614 | 0.0874 | 0.8377 | 0.8202 | 1 |