Ibrutinib KiNativ -- single dose experiment - Dataset (ID:20214)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| Ibrutinib | BCWM.1 | DNAPK | EHPFLVKGGEDLR | ATP | 40.00733586 | 1 | uM |
| Ibrutinib | BCWM.1 | DNAPK | KGGSWIQEINVAEK | ATP | 20.7626656 | 1 | uM |
| Ibrutinib | BCWM.1 | eEF2K | YIKYNSNSGFVR | ATP | 9.247436299 | 1 | uM |
| Ibrutinib | BCWM.1 | EPHB2 | FLEDDTSDPTYTSALGGKIPIR | Activation Loop | -13.84359152 | 1 | uM |
| Ibrutinib | BCWM.1 | MK03 | DLKPSNLLINTTCDLK | Lys2 | 11.91169046 | 1 | uM |
| Ibrutinib | BCWM.1 | Erk5 | DLKPSNLLVNENCELK | Lys2 | 19.32499308 | 1 | uM |
| Ibrutinib | BCWM.1 | FER | TSVAVKTCKEDLPQELK | Lys1 | 2.802692575 | 1 | uM |
| Ibrutinib | BCWM.1 | FES | LRADNTLVAVKSCR | Lys1 | -7.117814968 | 1 | uM |
| Ibrutinib | BCWM.1 | FGR | LIKDDEYNPCQGSKFPIK | Activation Loop | 73.81381667 | 1 | uM |
| Ibrutinib | BCWM.1 | FRAP1 | IQSIAPSLQVITSKQRPR | ATP | 12.08254388 | 1 | uM |
| Ibrutinib | BCWM.1 | FYN,SRC,YES | QGAKFPIKWTAPEAALYGR | Activation Loop | 22.58878067 | 1 | uM |
| Ibrutinib | BCWM.1 | GCK | DIKGANLLLTLQGDVK | Lys2 | -1.100183223 | 1 | uM |
| Ibrutinib | BCWM.1 | GCN2_domain2 | DLKPVNIFLDSDDHVK | Lys2 | -5.21921166 | 1 | uM |
| Ibrutinib | BCWM.1 | GSK3A | DIKPQNLLVDPDTAVLK | Lys2 | 10.9985253 | 1 | uM |
| Ibrutinib | BCWM.1 | GSK3B | DIKPQNLLLDPDTAVLK | Lys2 | 10.74352577 | 1 | uM |
| Ibrutinib | BCWM.1 | HPK1 | DIKGANILINDAGEVR | Lys2 | 8.152400611 | 1 | uM |
| Ibrutinib | BCWM.1 | IKKA | DLKPENIVLQDVGGK | Lys2 | -0.304730196 | 1 | uM |
| Ibrutinib | BCWM.1 | IKKB | DLKPENIVLQQGEQR | Lys2 | -6.412413441 | 1 | uM |
| Ibrutinib | BCWM.1 | IKKE | SGELVAVKVFNTTSYLRPR | Lys1 | -9.278395485 | 1 | uM |
| Ibrutinib | BCWM.1 | ILK | WQGNDIVVKVLK | Lys1 | -8.614846086 | 1 | uM |
| Ibrutinib | BCWM.1 | IRAK1 | AIQFLHQDSPSLIHGDIKSSNVLLDER | Lys2 | -25.21103032 | 1 | uM |
| Ibrutinib | BCWM.1 | IRAK4 | DIKSANILLDEAFTAK | Lys2 | -6.615440155 | 1 | uM |
| Ibrutinib | BCWM.1 | IRE1 | DLKPHNILISMPNAHGK | Lys2 | -15.99213778 | 1 | uM |
| Ibrutinib | BCWM.1 | ITPK1 | ESIFFNSHNVSKPESSSVLTELDKIEGVFERPSDEVIR | ATP | 16.25712664 | 1 | uM |
| Ibrutinib | BCWM.1 | JAK1 | QLASALSYLEDKDLVHGNVCTKNLLLAR | Other | 6.413468293 | 1 | uM |