Ibrutinib KiNativ -- single dose experiment - Dataset (ID:20214)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| Ibrutinib | BCWM.1 | CAMK1D | LFAVKCIPK | Lys1 | 9.317991024 | 1 | uM |
| Ibrutinib | BCWM.1 | CaMK2g | TSTQEYAAKIINTK | Lys1 | 5.984811925 | 1 | uM |
| Ibrutinib | MWCL.1 | CaMK2g | TSTQEYAAKIINTK | Lys1 | -5.159231787 | 1 | uM |
| Ibrutinib | MWCL.1 | CaMKK2 | DIKPSNLLVGEDGHIK | Lys2 | -3.023136542 | 1 | uM |
| Ibrutinib | BCWM.1 | CaMKK2 | DIKPSNLLVGEDGHIK | Lys2 | -22.22832801 | 1 | uM |
| Ibrutinib | MWCL.1 | CASK | ETGQQFAVKIVDVAK | Lys1 | 21.2690292 | 1 | uM |
| Ibrutinib | BCWM.1 | CASK | ETGQQFAVKIVDVAK | Lys1 | -0.612279673 | 1 | uM |
| Ibrutinib | BCWM.1 | CDC2 | DLKPQNLLIDDKGTIK | Lys2 | 3.199679306 | 1 | uM |
| Ibrutinib | MWCL.1 | CDC2 | DLKPQNLLIDDKGTIK | Lys2 | 4.72216791 | 1 | uM |
| Ibrutinib | MWCL.1 | CDK11,CDK8 | DLKPANILVMGEGPER | Lys2 | -25.79545872 | 1 | uM |
| Ibrutinib | BCWM.1 | CDK11,CDK8 | DLKPANILVMGEGPER | Lys2 | -23.27082009 | 1 | uM |
| Ibrutinib | MWCL.1 | CDK14 | LVALKVIR | Lys1 | 5.479239804 | 1 | uM |
| Ibrutinib | BCWM.1 | CDK14 | LVALKVIR | Lys1 | -8.300309889 | 1 | uM |
| Ibrutinib | MWCL.1 | CDK16 | SKLTDNLVALKEIR | Lys1 | -2.202969283 | 1 | uM |
| Ibrutinib | BCWM.1 | CDK16 | SKLTDNLVALKEIR | Lys1 | -26.55786151 | 1 | uM |
| Ibrutinib | BCWM.1 | CDK2 | DLKPQNLLINTEGAIK | Lys2 | -0.014042983 | 1 | uM |
| Ibrutinib | MWCL.1 | CDK2 | DLKPQNLLINTEGAIK | Lys2 | -0.986909811 | 1 | uM |
| Ibrutinib | BCWM.1 | CDK4 | DLKPENILVTSGGTVK | Lys2 | 5.962551436 | 1 | uM |
| Ibrutinib | MWCL.1 | CDK4 | DLKPENILVTSGGTVK | Lys2 | -5.399760136 | 1 | uM |
| Ibrutinib | BCWM.1 | CDK5 | DLKPQNLLINR | Lys2 | 9.033123773 | 1 | uM |
| Ibrutinib | MWCL.1 | CDK5 | DLKPQNLLINR | Lys2 | -10.15079399 | 1 | uM |
| Ibrutinib | BCWM.1 | CDK6 | DLKPQNILVTSSGQIK | Lys2 | -3.222110579 | 1 | uM |
| Ibrutinib | MWCL.1 | CDK6 | DLKPQNILVTSSGQIK | Lys2 | 7.22720664 | 1 | uM |
| Ibrutinib | BCWM.1 | CDK7 | DLKPNNLLLDENGVLK | Lys2 | 0.668563166 | 1 | uM |
| Ibrutinib | MWCL.1 | CDK7 | DLKPNNLLLDENGVLK | Lys2 | 2.518030866 | 1 | uM |