Ibrutinib KiNativ -- single dose experiment - Dataset (ID:20214)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
Ibrutinib MWCL.1 ZC1/HGK,ZC2/TNIK,ZC3/MINK
DIKGQNVLLTENAEVK
Lys2
-2.178793166
1
uM
Ibrutinib MWCL.1 ZC2/TNIK
TGQLAAIKVMDVTGDEEEEIKQEINMLKK
Lys1
-11.51803213
1
uM
Ibrutinib BCWM.1 ZC2/TNIK
TGQLAAIKVMDVTGDEEEEIKQEINMLKK
Lys1
-51.1480675
1
uM