Ibrutinib KiNativ -- single dose experiment - Dataset (ID:20214)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| Ibrutinib | BCWM.1 | NEK8 | DLKTQNILLDK | Lys2 | -15.33883097 | 1 | uM |
| Ibrutinib | MWCL.1 | NEK8 | DLKTQNILLDK | Lys2 | -10.81498066 | 1 | uM |
| Ibrutinib | BCWM.1 | NEK9 | DIKTLNIFLTK | Lys2 | 8.326033968 | 1 | uM |
| Ibrutinib | MWCL.1 | NEK9 | DIKTLNIFLTK | Lys2 | -0.237961412 | 1 | uM |
| Ibrutinib | MWCL.1 | OSR1 | DVKAGNILLGEDGSVQIADFGVSAFLATGGDITR | Lys2 | -5.216130694 | 1 | uM |
| Ibrutinib | BCWM.1 | OSR1 | DVKAGNILLGEDGSVQIADFGVSAFLATGGDITR | Lys2 | -1.255029683 | 1 | uM |
| Ibrutinib | MWCL.1 | p38a | DLKPSNLAVNEDCELK | Lys2 | -7.815671346 | 1 | uM |
| Ibrutinib | BCWM.1 | p38a | DLKPSNLAVNEDCELK | Lys2 | 11.12523953 | 1 | uM |
| Ibrutinib | BCWM.1 | p38d,p38g | DLKPGNLAVNEDCELK | Lys2 | 0.981795646 | 1 | uM |
| Ibrutinib | MWCL.1 | p38d,p38g | DLKPGNLAVNEDCELK | Lys2 | -15.19530384 | 1 | uM |
| Ibrutinib | BCWM.1 | PAN3 | VMDPTKILITGK | ATP | -19.88546356 | 1 | uM |
| Ibrutinib | MWCL.1 | PAN3 | VMDPTKILITGK | ATP | -27.71690181 | 1 | uM |
| Ibrutinib | MWCL.1 | PCTAIRE2,PCTAIRE3 | SKLTENLVALKEIR | Lys1 | 7.894332648 | 1 | uM |
| Ibrutinib | BCWM.1 | PCTAIRE2,PCTAIRE3 | SKLTENLVALKEIR | Lys1 | -14.73329296 | 1 | uM |
| Ibrutinib | BCWM.1 | PDK1 | EYAIKILEK | Lys1 | -26.37271999 | 1 | uM |
| Ibrutinib | MWCL.1 | PDK1 | EYAIKILEK | Lys1 | 21.2586975 | 1 | uM |
| Ibrutinib | BCWM.1 | PEK | DLKPSNIFFTMDDVVK | Lys2 | -23.81656725 | 1 | uM |
| Ibrutinib | MWCL.1 | PEK | DLKPSNIFFTMDDVVK | Lys2 | -31.61111339 | 1 | uM |
| Ibrutinib | BCWM.1 | PHKg2 | ATGHEFAVKIMEVTAER | Lys1 | -23.59607344 | 1 | uM |
| Ibrutinib | MWCL.1 | PHKg2 | ATGHEFAVKIMEVTAER | Lys1 | ND | 1 | uM |
| Ibrutinib | BCWM.1 | PI42C | TLVIKEVSSEDIADMHSNLSNYHQYIVK | ATP | -37.02302597 | 1 | uM |
| Ibrutinib | MWCL.1 | PI42C | TLVIKEVSSEDIADMHSNLSNYHQYIVK | ATP | -11.91082052 | 1 | uM |
| Ibrutinib | BCWM.1 | PI4KA,PI4KAP2 | SGTPMQSAAKAPYLAK | ATP | -19.55661054 | 1 | uM |
| Ibrutinib | MWCL.1 | PI4KA,PI4KAP2 | SGTPMQSAAKAPYLAK | ATP | -28.9504086 | 1 | uM |
| Ibrutinib | BCWM.1 | PI4KB | VPHTQAVVLNSKDK | ATP | -2.264791249 | 1 | uM |