Ibrutinib KiNativ -- single dose experiment - Dataset (ID:20214)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| Ibrutinib | BCWM.1 | M3K2,MAP3K3 | DIKGANILR | Lys2 | -12.68497138 | 1 | uM |
| Ibrutinib | BCWM.1 | M3K6 | DIKGDNVLINTFSGLLK | Lys2 | -18.14146781 | 1 | uM |
| Ibrutinib | BCWM.1 | MAP3K4 | DIKGANIFLTSSGLIK | Lys2 | -6.705973934 | 1 | uM |
| Ibrutinib | BCWM.1 | MAP3K5 | DIKGDNVLINTYSGVLK | Lys2 | 9.414089745 | 1 | uM |
| Ibrutinib | BCWM.1 | MARK2,MARK3 | DLKAENLLLDADMNIK | Lys2 | -14.37963599 | 1 | uM |
| Ibrutinib | BCWM.1 | MARK4 | DLKAENLLLDAEANIK | Lys2 | -11.00743851 | 1 | uM |
| Ibrutinib | BCWM.1 | MELK | DLKPENLLFDEYHK | Lys2 | -6.492711736 | 1 | uM |
| Ibrutinib | BCWM.1 | MAST1,MAST2 | DLKPDNLLITSMGHIK | Lys2 | -14.88979109 | 1 | uM |
| Ibrutinib | BCWM.1 | MAST3 | DLKPDNLLITSLGHIK | Lys2 | 7.95713657 | 1 | uM |
| Ibrutinib | MWCL.1 | LOK | DLKAGNVLMTLEGDIR | Lys2 | -31.7274951 | 1 | uM |
| Ibrutinib | BCWM.1 | NEK2 | DLKPANVFLDGK | Lys2 | 20.31739372 | 1 | uM |
| Ibrutinib | BCWM.1 | MLK3 | DLKSNNILLLQPIESDDMEHK | Lys2 | -22.45540747 | 1 | uM |
| Ibrutinib | BCWM.1 | MLK4 | DLKSSNILLLEK | Lys2 | 5.573785495 | 1 | uM |
| Ibrutinib | MWCL.1 | STK33 | DLKLENIMVK | Lys2 | -14.27502556 | 1 | uM |
| Ibrutinib | BCWM.1 | MSK1_domain1 | DIKLENILLDSNGHVVLTDFGLSK | Lys2 | 24.89837907 | 1 | uM |
| Ibrutinib | BCWM.1 | MSK2 domain1 | DLKLENVLLDSEGHIVLTDFGLSK | Lys2 | 40.22148406 | 1 | uM |
| Ibrutinib | BCWM.1 | RSK2 domain1 | DLKPENILLDEEGHIKLTDFGLSKESIDHEK | Lys2 | 20.13948334 | 1 | uM |
| Ibrutinib | BCWM.1 | STK33 | DLKLENIMVK | Lys2 | -32.70330347 | 1 | uM |
| Ibrutinib | BCWM.1 | MST3 | DIKAANVLLSEHGEVK | Lys2 | -9.956864462 | 1 | uM |
| Ibrutinib | MWCL.1 | CDK4 | DLKPENILVTSGGTVK | Lys2 | -5.399760136 | 1 | uM |
| Ibrutinib | BCWM.1 | MST4,YSK1 | DIKAANVLLSEQGDVK | Lys2 | -6.360178382 | 1 | uM |
| Ibrutinib | BCWM.1 | MYO3A,MYO3B | DVKGNNILLTTEGGVK | Lys2 | 7.942997988 | 1 | uM |
| Ibrutinib | BCWM.1 | NDR1 | DIKPDNLLLDSK | Lys2 | -1.353280454 | 1 | uM |
| Ibrutinib | BCWM.1 | NDR2 | DIKPDNLLLDAK | Lys2 | 1.201292359 | 1 | uM |
| Ibrutinib | BCWM.1 | NEK1 | DIKSQNIFLTK | Lys2 | -2.29771958 | 1 | uM |