Ibrutinib KiNativ -- single dose experiment - Dataset (ID:20214)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
Ibrutinib MWCL.1 STK33
DLKLENIMVK
Lys2
-14.27502556
1
uM
Ibrutinib MWCL.1 TYK2(Kin.Dom.2)
IGDFGLAKAVPEGHEYYR
Activation Loop
1.07145223
1
uM
Ibrutinib MWCL.1 Wnk1,Wnk2
GSFKTVYK
ATP Loop
6.431224998
1
uM