Ibrutinib KiNativ -- single dose experiment - Dataset (ID:20214)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| Ibrutinib | BCWM.1 | ARAF | DLKSNNIFLHEGLTVK | Lys2 | 0.09851812 | 1 | uM |
| Ibrutinib | BCWM.1 | ATR | FYIMMCKPK | ATP | -28.87734455 | 1 | uM |
| Ibrutinib | BCWM.1 | AurA | FILALKVLFK | Lys1 | 10.83507824 | 1 | uM |
| Ibrutinib | BCWM.1 | AurB | SHFIVALKVLFK | Lys1 | 5.086064352 | 1 | uM |
| Ibrutinib | BCWM.1 | BARK1 | DLKPANILLDEHGHVR | Lys2 | -16.279379 | 1 | uM |
| Ibrutinib | BCWM.1 | BRAF | DLKSNNIFLHEDLTVK | Lys2 | -15.53527116 | 1 | uM |
| Ibrutinib | BCWM.1 | BTK | YVLDDEYTSSVGSKFPVR | Activation Loop | 97.34431584 | 1 | uM |
| Ibrutinib | BCWM.1 | CAMK1D | LFAVKCIPK | Lys1 | 9.317991024 | 1 | uM |
| Ibrutinib | BCWM.1 | CaMK2g | TSTQEYAAKIINTK | Lys1 | 5.984811925 | 1 | uM |
| Ibrutinib | BCWM.1 | CaMKK2 | DIKPSNLLVGEDGHIK | Lys2 | -22.22832801 | 1 | uM |
| Ibrutinib | BCWM.1 | CASK | ETGQQFAVKIVDVAK | Lys1 | -0.612279673 | 1 | uM |
| Ibrutinib | BCWM.1 | CDC2 | DLKPQNLLIDDKGTIK | Lys2 | 3.199679306 | 1 | uM |
| Ibrutinib | BCWM.1 | CDK11,CDK8 | DLKPANILVMGEGPER | Lys2 | -23.27082009 | 1 | uM |
| Ibrutinib | BCWM.1 | CDK2 | DLKPQNLLINTEGAIK | Lys2 | -0.014042983 | 1 | uM |
| Ibrutinib | BCWM.1 | CDK4 | DLKPENILVTSGGTVK | Lys2 | 5.962551436 | 1 | uM |
| Ibrutinib | BCWM.1 | CDK5 | DLKPQNLLINR | Lys2 | 9.033123773 | 1 | uM |
| Ibrutinib | BCWM.1 | CDK6 | DLKPQNILVTSSGQIK | Lys2 | -3.222110579 | 1 | uM |
| Ibrutinib | BCWM.1 | CDK7 | DLKPNNLLLDENGVLK | Lys2 | 0.668563166 | 1 | uM |
| Ibrutinib | BCWM.1 | CDK9 | DMKAANVLITR | Lys2 | -36.25571353 | 1 | uM |
| Ibrutinib | BCWM.1 | CHK1 | DIKPENLLLDER | Lys2 | -18.34031487 | 1 | uM |
| Ibrutinib | BCWM.1 | CHK2 | DLKPENVLLSSQEEDCLIK | Lys2 | 8.060736198 | 1 | uM |
| Ibrutinib | BCWM.1 | KC1A | DIKPDNFLMGIGR | Lys2 | -31.76193819 | 1 | uM |
| Ibrutinib | BCWM.1 | CK2a2 | DVKPHNVMIDHQQK | Lys2 | -10.76125661 | 1 | uM |
| Ibrutinib | BCWM.1 | CSK | VSDFGLTKEASSTQDTGKLPVK | Activation Loop | 15.82121782 | 1 | uM |
| Ibrutinib | BCWM.1 | DGKA | IDPVPNTHPLLVFVNPKSGGK | ATP | ND | 1 | uM |