JNK-IN-8 KiNativ -- single dose experiment - Dataset (ID:20213)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
JNK-IN-8 | A-375 | NDR2 | DIkPDNLLLDAK | Lys2 | 14.7 | 1 | uM |
JNK-IN-8 | A-375 | NDR1 | DIkPDNLLLDSK | Lys2 | 5.8 | 1 | uM |
JNK-IN-8 | A-375 | CHK1 | DIkPENLLLDERDNLK | Lys2 | 8.7 | 1 | uM |
JNK-IN-8 | A-375 | AurA | DIkPENLLLGSAGELK | Lys2 | -8.0 | 1 | uM |
JNK-IN-8 | A-375 | IKKE,TBK1 | DIkPGNIMR | Lys2 | -24.5 | 1 | uM |
JNK-IN-8 | A-375 | LKB1 | DIkPGNLLLTTGGTLK | Lys2 | -20.1 | 1 | uM |
JNK-IN-8 | A-375 | GSK3B | DIkPQNLLLDPDTAVLK | Lys2 | -8.5 | 1 | uM |
JNK-IN-8 | A-375 | GSK3A | DIkPQNLLVDPDTAVLK | Lys2 | 10.6 | 1 | uM |
JNK-IN-8 | A-375 | MAP2K4 | DIkPSNILLDR | Lys2 | -12.0 | 1 | uM |
JNK-IN-8 | A-375 | IRAK4 | DIkSANILLDEAFTAK | Lys2 | 6.4 | 1 | uM |
JNK-IN-8 | A-375 | NEK1 | DIkSQNIFLTK | Lys2 | -12.1 | 1 | uM |
JNK-IN-8 | A-375 | NEK9 | DIkTLNIFLTK | Lys2 | -32.2 | 1 | uM |
JNK-IN-8 | A-375 | FER | DKTSVAVkTCKEDLPQELK | Lys1 | 13.9 | 1 | uM |
JNK-IN-8 | A-375 | MARK2,MARK3 | DLkAENLLLDADMNIK | Lys2 | 13.9 | 1 | uM |
JNK-IN-8 | A-375 | MARK1 | DLkAENLLLDGDMNIK | Lys2 | 8.9 | 1 | uM |
JNK-IN-8 | A-375 | SLK | DLkAGNILFTLDGDIK | Lys2 | 17.2 | 1 | uM |
JNK-IN-8 | A-375 | SLK | DLkAGNILFTLDGDIKLADFGVSAK | Lys2 | 3.2 | 1 | uM |
JNK-IN-8 | A-375 | LOK | DLkAGNVLMTLEGDIR | Lys2 | 2.8 | 1 | uM |
JNK-IN-8 | A-375 | Wnk1,Wnk2,Wnk3 | DLkCDNIFITGPTGSVK | Lys2 | 12.7 | 1 | uM |
JNK-IN-8 | A-375 | WNK4 | DLkCDNVFITGPTGSVK | Lys2 | 16.1 | 1 | uM |
JNK-IN-8 | A-375 | KPCT | DLkLDNILLDK | Lys2 | -19.5 | 1 | uM |
JNK-IN-8 | A-375 | PKN2 | DLkLDNLLLDTEGFVK | Lys2 | -7.3 | 1 | uM |
JNK-IN-8 | A-375 | CDK11,CDK8 | DLkPANILVMGEGPER | Lys2 | 0.4 | 1 | uM |
JNK-IN-8 | A-375 | MAST3 | DLkPDNLLITSLGHIK | Lys2 | 13.9 | 1 | uM |
JNK-IN-8 | A-375 | MAST1,MAST2 | DLkPDNLLITSMGHIK | Lys2 | -31.3 | 1 | uM |