JNK-IN-8 KiNativ -- single dose experiment - Dataset (ID:20213)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| JNK-IN-8 | A-375 | CDK14 | LVALkVIR | Lys1 | 38.1 | 1 | uM |
| JNK-IN-8 | A-375 | CDK16 | LTDNLVALkEIR | Lys1 | -9.0 | 1 | uM |
| JNK-IN-8 | A-375 | CDK2 | DLkPQNLLINTEGAIK | Lys2 | -9.0 | 1 | uM |
| JNK-IN-8 | A-375 | CDK2 | NKLTGEVVALkK | Lys1 | -3.8 | 1 | uM |
| JNK-IN-8 | A-375 | CDK4 | DLkPENILVTSGGTVK | Lys2 | -17.3 | 1 | uM |
| JNK-IN-8 | A-375 | CDK5 | NVLHRDLkPQNLLINR | Lys2 | 7.4 | 1 | uM |
| JNK-IN-8 | A-375 | CDK5 | NRETHEIVALkR | Lys1 | 3.3 | 1 | uM |
| JNK-IN-8 | A-375 | CDK6 | DLkPQNILVTSSGQIK | Lys2 | -20.9 | 1 | uM |
| JNK-IN-8 | A-375 | CDK7 | DLkPNNLLLDENGVLK | Lys2 | -2.9 | 1 | uM |
| JNK-IN-8 | A-375 | CDK9 | DMkAANVLITR | Lys2 | -34.1 | 1 | uM |
| JNK-IN-8 | A-375 | CHK1 | LSkGDGLEFK | Other | -38.8 | 1 | uM |
| JNK-IN-8 | A-375 | CHK1 | DIkPENLLLDERDNLK | Lys2 | 8.7 | 1 | uM |
| JNK-IN-8 | A-375 | CHK2 | VAIkIISK | Lys1 | -3.8 | 1 | uM |
| JNK-IN-8 | A-375 | CK1d,CK1e | DVkPDNFLMGLGKK | Lys2 | -21.8 | 1 | uM |
| JNK-IN-8 | A-375 | CK2a1 | GGPNIITLADIVkDPVSR | Protein Kinase Domain | -31.1 | 1 | uM |
| JNK-IN-8 | A-375 | CSK | VSDFGLTkEASSTQDTGK | Activation Loop | 23.4 | 1 | uM |
| JNK-IN-8 | A-375 | CSK | VSDFGLTkEASSTQDTGKLPVK | Activation Loop | 4.3 | 1 | uM |
| JNK-IN-8 | A-375 | DGKA | IDPVPNTHPLLVFVNPkSGGK | ATP | -25.9 | 1 | uM |
| JNK-IN-8 | A-375 | DMPK | DIkPDNILLDR | Lys2 | -3.2 | 1 | uM |
| JNK-IN-8 | A-375 | DNAPK | GHDEREHPFLVkGGEDLRQDQR | ATP | 10.5 | 1 | uM |
| JNK-IN-8 | A-375 | DNAPK | EHPFLVkGGEDLR | ATP | -19.3 | 1 | uM |
| JNK-IN-8 | A-375 | DNAPK | GHDEREHPFLVkGGEDLR | ATP | 34.9 | 1 | uM |
| JNK-IN-8 | A-375 | DNAPK | kGGSWIQEINVAEK | ATP | 12.8 | 1 | uM |
| JNK-IN-8 | A-375 | DNAPK | kGGSWIQEINVAEKNWYPR | ATP | 14.7 | 1 | uM |
| JNK-IN-8 | A-375 | eEF2K | YIkYNSNSGFVR | Protein Kinase Domain | -5.4 | 1 | uM |