JNK-IN-8 KiNativ -- single dose experiment - Dataset (ID:20213)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
JNK-IN-8 A-375 MAST2,MAST4
DLkPDNLLVTSMGHIK
Lys2
-8.9
1
uM
JNK-IN-8 A-375 MAP2K6
MCDFGISGYLVDSVAkTIDAGCKPYMAPER
Activation Loop
-8.9
1
uM
JNK-IN-8 A-375 p38d,p38g
DLkPGNLAVNEDCELK
Lys2
-8.9
1
uM
JNK-IN-8 A-375 MARK1
DLkAENLLLDGDMNIK
Lys2
8.9
1
uM
JNK-IN-8 A-375 CDK2
DLkPQNLLINTEGAIK
Lys2
-9.0
1
uM
JNK-IN-8 A-375 CDK16
LTDNLVALkEIR
Lys1
-9.0
1
uM
JNK-IN-8 A-375 GCN2_domain2
VQNKLDGCCYAVkR
Lys1
9.0
1
uM
JNK-IN-8 A-375 PIK3CA
RPLWLNWENPDIMSELLFQNNEIIFkNGDDLRQDMLTLQIIR
ATP
-9.2
1
uM
JNK-IN-8 A-375 KCC2D
CMKIPTGQEYAAkIINTK
Lys1
-9.2
1
uM
JNK-IN-8 A-375 NEK8
DLkTQNILLDK
Lys2
-9.6
1
uM
JNK-IN-8 A-375 MARK2
HILTGKEVAVkIIDKTQLNSSSLQK
Lys1
9.6
1
uM
JNK-IN-8 A-375 MAP2K5
DVkPSNMLVNTR
Lys2
-9.7
1
uM
JNK-IN-8 A-375 STLK5
YSVkVLPWLSPEVLQQNLQGYDAK
Activation Loop
9.7
1
uM
JNK-IN-8 A-375 JNK1,JNK2,JNK3
DLkPSNIVVK
Lys2
98.7
1
uM
JNK-IN-8 A-375 ZC2/TNIK
TGQLAAIkVMDVTGDEEEEIKQEINMLKK
Lys1
9.9
1
uM