OTSSP167 KiNativ -- single dose experiment - Dataset (ID:20209)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
OTSSP167 | MDA-MB-468 | DNAPK | KGGSWIQEINVAEK | ATP | >97 | 1 | uM |
OTSSP167 | MDA-MB-468 | DNAPK | EHPFLVKGGEDLR | ATP | 98.8 | 1 | uM |
OTSSP167 | MDA-MB-468 | eEF2K | YIKYNSNSGFVR | ATP | -2.3 | 1 | uM |
OTSSP167 | MDA-MB-468 | EGFR | LLGAEEKEYHAEGGKVPIK | Activation Loop | 29.0 | 1 | uM |
OTSSP167 | MDA-MB-468 | EphA1 | LLDDFDGTYETQGGKIPIR | Activation Loop | >97 | 1 | uM |
OTSSP167 | MDA-MB-468 | EPHA2 | VLEDDPEATYTTSGGKIPIR | Activation Loop | >98 | 1 | uM |
OTSSP167 | MDA-MB-468 | EPHB2 | FLEDDTSDPTYTSALGGKIPIR | Activation Loop | >96 | 1 | uM |
OTSSP167 | MDA-MB-468 | EPHB4 | FLEENSSDPTYTSSLGGKIPIR | Activation Loop | >95 | 1 | uM |
OTSSP167 | MDA-MB-468 | MK03 | DLKPSNLLINTTCDLK | Lys2 | 1.5 | 1 | uM |
OTSSP167 | MDA-MB-468 | FER | TSVAVKTCKEDLPQELK | Lys1 | 99.8 | 1 | uM |
OTSSP167 | MDA-MB-468 | FRAP1 | IQSIAPSLQVITSKQRPR | ATP | 92.1 | 1 | uM |
OTSSP167 | MDA-MB-468 | FYN,SRC,YES | QGAKFPIKWTAPEAALYGR | Activation Loop | 83.9 | 1 | uM |
OTSSP167 | MDA-MB-468 | GCK | DIKGANLLLTLQGDVK | Lys2 | 96.5 | 1 | uM |
OTSSP167 | MDA-MB-468 | GCN2_domain2 | DLKPVNIFLDSDDHVK | Lys2 | 90.9 | 1 | uM |
OTSSP167 | MDA-MB-468 | GSK3A | DIKPQNLLVDPDTAVLK | Lys2 | >99 | 1 | uM |
OTSSP167 | MDA-MB-468 | GSK3B | DIKPQNLLLDPDTAVLK | Lys2 | >99 | 1 | uM |
OTSSP167 | MDA-MB-468 | IKKA | DLKPENIVLQDVGGK | Lys2 | 5.2 | 1 | uM |
OTSSP167 | MDA-MB-468 | IKKB | DLKPENIVLQQGEQR | Lys2 | -12.0 | 1 | uM |
OTSSP167 | MDA-MB-468 | IKKE | SGELVAVKVFNTTSYLRPR | Lys1 | >93 | 1 | uM |
OTSSP167 | MDA-MB-468 | ILK | WQGNDIVVKVLK | Lys1 | 18.0 | 1 | uM |
OTSSP167 | MDA-MB-468 | IRAK1 | AIQFLHQDSPSLIHGDIKSSNVLLDER | Lys2 | 83.1 | 1 | uM |
OTSSP167 | MDA-MB-468 | IRAK4 | DIKSANILLDEAFTAK | Lys2 | 97.3 | 1 | uM |
OTSSP167 | MDA-MB-468 | IRE1 | DLKPHNILISMPNAHGK | Lys2 | 68.7 | 1 | uM |
OTSSP167 | MDA-MB-468 | ITPK1 | ESIFFNSHNVSKPESSSVLTELDKIEGVFERPSDEVIR | ATP | 25.7 | 1 | uM |
OTSSP167 | MDA-MB-468 | JAK1 | QLASALSYLEDKDLVHGNVCTKNLLLAR | Protein Kinase Domain | 41.7 | 1 | uM |