OTSSP167 KiNativ -- single dose experiment - Dataset (ID:20209)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| OTSSP167 | MDA-MB-468 | CaMK2g | TSTQEYAAKIINTK | Lys1 | 87.9 | 1 | uM |
| OTSSP167 | MDA-MB-468 | FER | TSVAVKTCKEDLPQELK | Lys1 | 99.8 | 1 | uM |
| OTSSP167 | MDA-MB-468 | ACK | TVSVAVKCLKPDVLSQPEAMDDFIR | Lys1 | 72.3 | 1 | uM |
| OTSSP167 | MDA-MB-468 | YES | VAIKTLKPGTMMPEAFLQEAQIMK | Lys1 | >88 | 1 | uM |
| OTSSP167 | MDA-MB-468 | EPHA2 | VLEDDPEATYTTSGGKIPIR | Activation Loop | >98 | 1 | uM |
| OTSSP167 | MDA-MB-468 | RSKL1_domain1 | VLGVIDKVLLVMDTR | ATP | -41.3 | 1 | uM |
| OTSSP167 | MDA-MB-468 | PKN1 | VLLSEFRPSGELFAIKALK | Lys1 | 95.8 | 1 | uM |
| OTSSP167 | MDA-MB-468 | PAN3 | VMDPTKILITGK | ATP | -21.3 | 1 | uM |
| OTSSP167 | MDA-MB-468 | PI4KB | VPHTQAVVLNSKDK | ATP | >98 | 1 | uM |
| OTSSP167 | MDA-MB-468 | CSK | VSDFGLTKEASSTQDTGKLPVK | Activation Loop | 92.1 | 1 | uM |
| OTSSP167 | MDA-MB-468 | MLTK | WISQDKEVAVKK | Lys1 | >98 | 1 | uM |
| OTSSP167 | MDA-MB-468 | ILK | WQGNDIVVKVLK | Lys1 | 18.0 | 1 | uM |
| OTSSP167 | MDA-MB-468 | CLK3 | YEIVGNLGEGTFGKVVECLDHAR | ATP Loop | 98.4 | 1 | uM |
| OTSSP167 | MDA-MB-468 | eEF2K | YIKYNSNSGFVR | ATP | -2.3 | 1 | uM |
| OTSSP167 | MDA-MB-468 | TLK1 | YLNEIKPPIIHYDLKPGNILLVDGTACGEIK | Lys2 | 53.7 | 1 | uM |
| OTSSP167 | MDA-MB-468 | TLK1/2 | YLNEIKPPIIHYDLKPGNILLVNGTACGEIK | Lys2 | 16.7 | 1 | uM |
| OTSSP167 | MDA-MB-468 | MK09 | YQQLKPIGSGAQGIVCAAFDTVLGINVAVKK | Lys1 | 44.1 | 1 | uM |
| OTSSP167 | MDA-MB-468 | STLK5 | YSVKVLPWLSPEVLQQNLQGYDAK | Activation Loop | 83.5 | 1 | uM |