OTSSP167 KiNativ -- single dose experiment - Dataset (ID:20209)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| OTSSP167 | MDA-MB-468 | SMG1 | DTVTIHSVGGTITILPTKTKPK | ATP | 98.1 | 1 | uM |
| OTSSP167 | MDA-MB-468 | SNRK | DLKPENVVFFEK | Lys2 | 12.8 | 1 | uM |
| OTSSP167 | MDA-MB-468 | SRPK1 | IIHTDIKPENILLSVNEQYIR | Lys2 | 86.8 | 1 | uM |
| OTSSP167 | MDA-MB-468 | SRPK1/2 | FVAMKVVK | Lys1 | 72.8 | 1 | uM |
| OTSSP167 | MDA-MB-468 | STLK5 | YSVKVLPWLSPEVLQQNLQGYDAK | Activation Loop | 83.5 | 1 | uM |
| OTSSP167 | MDA-MB-468 | SYK | ISDFGLSKALR | Activation Loop | 91.6 | 1 | uM |
| OTSSP167 | MDA-MB-468 | TAO1,TAOK3 | DIKAGNILLTEPGQVK | Lys2 | >99 | 1 | uM |
| OTSSP167 | MDA-MB-468 | TAOK2 | DVKAGNILLSEPGLVK | Lys2 | >97 | 1 | uM |
| OTSSP167 | MDA-MB-468 | TBK1 | TGDLFAIKVFNNISFLRPVDVQMR | Lys1 | >90 | 1 | uM |
| OTSSP167 | MDA-MB-468 | TLK1 | YLNEIKPPIIHYDLKPGNILLVDGTACGEIK | Lys2 | 53.7 | 1 | uM |
| OTSSP167 | MDA-MB-468 | TLK1/2 | YLNEIKPPIIHYDLKPGNILLVNGTACGEIK | Lys2 | 16.7 | 1 | uM |
| OTSSP167 | MDA-MB-468 | TNK1 | SVPVAVKSLR | Lys1 | >95 | 1 | uM |
| OTSSP167 | MDA-MB-468 | TYK2(Kin.Dom.2) | IGDFGLAKAVPEGHEYYR | Activation Loop | 88.4 | 1 | uM |
| OTSSP167 | MDA-MB-468 | ULK1 | DLKPQNILLSNPAGR | Lys2 | -64.2 | 1 | uM |
| OTSSP167 | MDA-MB-468 | ULK3 | NISHLDLKPQNILLSSLEKPHLK | Lys2 | 75.3 | 1 | uM |
| OTSSP167 | MDA-MB-468 | Wnk1,Wnk2,Wnk3 | DLKCDNIFITGPTGSVK | Lys2 | 12.6 | 1 | uM |
| OTSSP167 | MDA-MB-468 | YES | VAIKTLKPGTMMPEAFLQEAQIMK | Lys1 | >88 | 1 | uM |
| OTSSP167 | MDA-MB-468 | ZC1/HGK,ZC2/TNIK,ZC3/MINK | DIKGQNVLLTENAEVK | Lys2 | >98 | 1 | uM |