OTSSP167 KiNativ -- single dose experiment - Dataset (ID:20209)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
OTSSP167 | MDA-MB-468 | LOK | DLKAGNVLMTLEGDIR | Lys2 | 98.0 | 1 | uM |
OTSSP167 | MDA-MB-468 | MAP2K1 | IMHRDVKPSNILVNSR | Lys2 | 98.0 | 1 | uM |
OTSSP167 | MDA-MB-468 | MST4,YSK1 | DIKAANVLLSEQGDVK | Lys2 | 98.0 | 1 | uM |
OTSSP167 | MDA-MB-468 | SMG1 | DTVTIHSVGGTITILPTKTKPK | ATP | 98.1 | 1 | uM |
OTSSP167 | MDA-MB-468 | AMPKa1,AMPKa2 | DLKPENVLLDAHMNAK | Lys2 | 98.2 | 1 | uM |
OTSSP167 | MDA-MB-468 | RSK1 domain1 | DLKPENILLDEEGHIKLTDFGLSKEAIDHEK | Lys2 | 98.4 | 1 | uM |
OTSSP167 | MDA-MB-468 | CLK3 | YEIVGNLGEGTFGKVVECLDHAR | ATP Loop | 98.4 | 1 | uM |
OTSSP167 | MDA-MB-468 | MST3 | DIKAANVLLSEHGEVK | Lys2 | 98.4 | 1 | uM |
OTSSP167 | MDA-MB-468 | RSK1,RSK2,RSK3_domain1 | DLKPENILLDEEGHIK | Lys2 | 98.5 | 1 | uM |
OTSSP167 | MDA-MB-468 | MAP2K1,MAP2K2 | DVKPSNILVNSR | Lys2 | 98.5 | 1 | uM |
OTSSP167 | MDA-MB-468 | CDK2 | DLKPQNLLINTEGAIK | Lys2 | 98.7 | 1 | uM |
OTSSP167 | MDA-MB-468 | DNAPK | EHPFLVKGGEDLR | ATP | 98.8 | 1 | uM |
OTSSP167 | MDA-MB-468 | AurB | SHFIVALKVLFK | Lys1 | >99 | 1 | uM |
OTSSP167 | MDA-MB-468 | MST2 | ESGQVVAIKQVPVESDLQEIIK | Lys1 | >99 | 1 | uM |
OTSSP167 | MDA-MB-468 | TAO1,TAOK3 | DIKAGNILLTEPGQVK | Lys2 | >99 | 1 | uM |
OTSSP167 | MDA-MB-468 | GSK3B | DIKPQNLLLDPDTAVLK | Lys2 | >99 | 1 | uM |
OTSSP167 | MDA-MB-468 | GSK3A | DIKPQNLLVDPDTAVLK | Lys2 | >99 | 1 | uM |
OTSSP167 | MDA-MB-468 | FER | TSVAVKTCKEDLPQELK | Lys1 | 99.8 | 1 | uM |