OTSSP167 KiNativ -- single dose experiment - Dataset (ID:20209)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
OTSSP167 | MDA-MB-468 | NEK9 | DIKTLNIFLTK | Lys2 | 50.1 | 1 | uM |
OTSSP167 | MDA-MB-468 | KHS1 | NVHTGELAAVKIIK | Lys1 | 51.5 | 1 | uM |
OTSSP167 | MDA-MB-468 | IKKA | DLKPENIVLQDVGGK | Lys2 | 5.2 | 1 | uM |
OTSSP167 | MDA-MB-468 | TLK1 | YLNEIKPPIIHYDLKPGNILLVDGTACGEIK | Lys2 | 53.7 | 1 | uM |
OTSSP167 | MDA-MB-468 | CDK13 | DIKCSNILLNNR | Lys2 | 56.1 | 1 | uM |
OTSSP167 | MDA-MB-468 | NDR2 | DIKPDNLLLDAK | Lys2 | 58.1 | 1 | uM |
OTSSP167 | MDA-MB-468 | NEK4 | DLKTQNVFLTR | Lys2 | 58.2 | 1 | uM |
OTSSP167 | MDA-MB-468 | CRK7 | DIKCSNILLNNSGQIK | Lys2 | 59.6 | 1 | uM |
OTSSP167 | MDA-MB-468 | OSR1 | DVKAGNILLGEDGSVQIADFGVSAFLATGGDITR | Lys2 | 60.5 | 1 | uM |
OTSSP167 | MDA-MB-468 | NEK2 | DLKPANVFLDGK | Lys2 | 61.1 | 1 | uM |
OTSSP167 | MDA-MB-468 | KS6B1 | DLKPENIMLNHQGHVK | Lys2 | 62.1 | 1 | uM |
OTSSP167 | MDA-MB-468 | MARK2,MARK3 | DLKAENLLLDADMNIK | Lys2 | 63.0 | 1 | uM |
OTSSP167 | MDA-MB-468 | ULK1 | DLKPQNILLSNPAGR | Lys2 | -64.2 | 1 | uM |
OTSSP167 | MDA-MB-468 | PKMYT1 | DTLLALAHLHSQGLVHLDVKPANIFLGPR | Lys2 | 65.8 | 1 | uM |
OTSSP167 | MDA-MB-468 | NDR1 | DIKPDNLLLDSK | Lys2 | 68.4 | 1 | uM |
OTSSP167 | MDA-MB-468 | IRE1 | DLKPHNILISMPNAHGK | Lys2 | 68.7 | 1 | uM |
OTSSP167 | MDA-MB-468 | PEK | DLKPSNIFFTMDDVVK | Lys2 | 70.9 | 1 | uM |
OTSSP167 | MDA-MB-468 | ACK | TVSVAVKCLKPDVLSQPEAMDDFIR | Lys1 | 72.3 | 1 | uM |
OTSSP167 | MDA-MB-468 | SRPK1/2 | FVAMKVVK | Lys1 | 72.8 | 1 | uM |
OTSSP167 | MDA-MB-468 | MLKL | APVAIKVFK | Lys1 | 73.3 | 1 | uM |
OTSSP167 | MDA-MB-468 | PRPK | FLSGLELVKQGAEAR | ATP Loop | 73.5 | 1 | uM |
OTSSP167 | MDA-MB-468 | ULK3 | NISHLDLKPQNILLSSLEKPHLK | Lys2 | 75.3 | 1 | uM |
OTSSP167 | MDA-MB-468 | CAMK1D | LFAVKCIPK | Lys1 | 75.8 | 1 | uM |
OTSSP167 | MDA-MB-468 | PHKg2 | ATGHEFAVKIMEVTAER | Lys1 | 75.9 | 1 | uM |
OTSSP167 | MDA-MB-468 | BRAF | DLKSNNIFLHEDLTVK | Lys2 | 7.6 | 1 | uM |