QL-XII-47 KiNativ -- single dose experiment - Dataset (ID:20205)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| QL-XII-47 | MWCL.1 | PHKg2 | ATGHEFAVKIMEVTAER | Lys1 | ND | 1 | uM |
| QL-XII-47 | MWCL.1 | EPHB2 | FLEDDTSDPTYTSALGGKIPIR | Activation Loop | ND | 1 | uM |
| QL-XII-47 | MWCL.1 | BLK | IIDSEYTAQEGAKFPIK | Activation Loop | ND | 1 | uM |
| QL-XII-47 | BCWM.1 | DGKA | IDPVPNTHPLLVFVNPKSGGK | ATP | ND | 1 | uM |
| QL-XII-47 | MWCL.1 | M3K6 | DIKGDNVLINTFSGLLK | Lys2 | ND | 1 | uM |
| QL-XII-47 | MWCL.1 | RSK4 domain1 | DLKPENILLDEIGHIK | Lys2 | ND | 1 | uM |
| QL-XII-47 | MWCL.1 | MLK4 | DLKSSNILLLEK | Lys2 | ND | 1 | uM |
| QL-XII-47 | MWCL.1 | EPHB1 | YLQDDTSDPTYTSSLGGKIPVR | Activation Loop | ND | 1 | uM |
| QL-XII-47 | BCWM.1 | STLK6 | HTPTGTLVTIKITNLENCNEER | Lys1 | ND | 1 | uM |
| QL-XII-47 | MWCL.1 | SYK | ISDFGLSKALR | Activation Loop | 9.937407948 | 1 | uM |
| QL-XII-47 | MWCL.1 | CK2a2 | DVKPHNVMIDHQQK | Lys2 | -9.931851645 | 1 | uM |
| QL-XII-47 | MWCL.1 | NEK3 | SKNIFLTQNGK | Activation Loop | 9.919741065 | 1 | uM |
| QL-XII-47 | MWCL.1 | MK03 | DLKPSNLLINTTCDLK | Lys2 | -9.820784106 | 1 | uM |
| QL-XII-47 | MWCL.1 | MAP3K5 | DIKGDNVLINTYSGVLK | Lys2 | -9.625870933 | 1 | uM |
| QL-XII-47 | BCWM.1 | MARK3 | EVAIKIIDKTQLNPTSLQK | Lys1 | -9.506780432 | 1 | uM |
| QL-XII-47 | BCWM.1 | NEK8 | DLKTQNILLDK | Lys2 | 9.444227339 | 1 | uM |
| QL-XII-47 | MWCL.1 | JAK1_domain2 | IGDFGLTKAIETDKEYYTVK | Activation Loop | -9.341503001 | 1 | uM |
| QL-XII-47 | BCWM.1 | CDK4 | DLKPENILVTSGGTVK | Lys2 | -9.229049081 | 1 | uM |
| QL-XII-47 | MWCL.1 | MAP3K1 | DVKGANLLIDSTGQR | Lys2 | 9.175244255 | 1 | uM |
| QL-XII-47 | BCWM.1 | RIPK3 | DLKPSNVLLDPELHVK | Lys2 | -9.173875348 | 1 | uM |
| QL-XII-47 | MWCL.1 | SGK3 | FYAVKVLQK | Lys1 | 9.129996049 | 1 | uM |
| QL-XII-47 | BCWM.1 | MK11 | QELNKTVWEVPQR | Other | 9.053676509 | 1 | uM |
| QL-XII-47 | MWCL.1 | PAN3 | VMDPTKILITGK | ATP | 9.049225166 | 1 | uM |
| QL-XII-47 | BCWM.1 | FYV1 | GGKSGAAFYATEDDRFILK | ATP | 9.038475869 | 1 | uM |
| QL-XII-47 | BCWM.1 | MST2 | ESGQVVAIKQVPVESDLQEIIK | Lys1 | 9.022179848 | 1 | uM |