QL-XII-47 KiNativ -- single dose experiment - Dataset (ID:20205)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
QL-XII-47 | BCWM.1 | CASK | ETGQQFAVKIVDVAK | Lys1 | 32.90610469 | 1 | uM |
QL-XII-47 | BCWM.1 | CDK9 | DMKAANVLITR | Lys2 | 11.68818243 | 1 | uM |
QL-XII-47 | BCWM.1 | AurA | FILALKVLFK | Lys1 | 19.31283508 | 1 | uM |
QL-XII-47 | BCWM.1 | CaMKK2 | DIKPSNLLVGEDGHIK | Lys2 | 11.88734459 | 1 | uM |
QL-XII-47 | BCWM.1 | CDK4 | DLKPENILVTSGGTVK | Lys2 | -9.229049081 | 1 | uM |
QL-XII-47 | BCWM.1 | CDK7 | DLKPNNLLLDENGVLK | Lys2 | 15.31231831 | 1 | uM |
QL-XII-47 | BCWM.1 | ACK | TVSVAVKCLKPDVLSQPEAMDDFIR | Lys1 | 16.75144083 | 1 | uM |
QL-XII-47 | BCWM.1 | ATR | FYIMMCKPK | ATP | 0.044349501 | 1 | uM |
QL-XII-47 | BCWM.1 | BRAF | DLKSNNIFLHEDLTVK | Lys2 | 17.78977881 | 1 | uM |
QL-XII-47 | BCWM.1 | CaMK2g | TSTQEYAAKIINTK | Lys1 | 4.50076179 | 1 | uM |
QL-XII-47 | BCWM.1 | CDK11,CDK8 | DLKPANILVMGEGPER | Lys2 | 14.74034939 | 1 | uM |
QL-XII-47 | BCWM.1 | CDK2 | DLKPQNLLINTEGAIK | Lys2 | -1.556399301 | 1 | uM |
QL-XII-47 | BCWM.1 | CDK5 | DLKPQNLLINR | Lys2 | 4.004453656 | 1 | uM |
QL-XII-47 | BCWM.1 | CDK6 | DLKPQNILVTSSGQIK | Lys2 | -0.544166997 | 1 | uM |
QL-XII-47 | BCWM.1 | ABL,ARG | LMTGDTYTAHAGAKFPIK | Activation Loop | -4.884271122 | 1 | uM |
QL-XII-47 | BCWM.1 | ABL,ARG | YSLTVAVKTLKEDTMEVEEFLK | Lys1 | 23.94636209 | 1 | uM |
QL-XII-47 | BCWM.1 | AMPKa1,AMPKa2 | DLKPENVLLDAHMNAK | Lys2 | 18.43323382 | 1 | uM |
QL-XII-47 | BCWM.1 | ARAF | DLKSNNIFLHEGLTVK | Lys2 | 4.534711447 | 1 | uM |
QL-XII-47 | BCWM.1 | AurB | SHFIVALKVLFK | Lys1 | 7.861261294 | 1 | uM |
QL-XII-47 | BCWM.1 | BARK1 | DLKPANILLDEHGHVR | Lys2 | -22.46332421 | 1 | uM |
QL-XII-47 | BCWM.1 | BTK | YVLDDEYTSSVGSKFPVR | Activation Loop | 70.55327861 | 1 | uM |
QL-XII-47 | BCWM.1 | CAMK1D | LFAVKCIPK | Lys1 | 0.033712822 | 1 | uM |
QL-XII-47 | BCWM.1 | CDC2 | DLKPQNLLIDDKGTIK | Lys2 | -11.32754424 | 1 | uM |
QL-XII-47 | BCWM.1 | CHK2 | DLKPENVLLSSQEEDCLIK | Lys2 | 1.250240618 | 1 | uM |
QL-XII-47 | BCWM.1 | CHK1 | DIKPENLLLDER | Lys2 | 2.996204004 | 1 | uM |