QL-XII-47 KiNativ -- single dose experiment - Dataset (ID:20205)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
QL-XII-47 BCWM.1 CASK
ETGQQFAVKIVDVAK
Lys1
32.90610469
1
uM
QL-XII-47 BCWM.1 CDK9
DMKAANVLITR
Lys2
11.68818243
1
uM
QL-XII-47 BCWM.1 AurA
FILALKVLFK
Lys1
19.31283508
1
uM
QL-XII-47 BCWM.1 CaMKK2
DIKPSNLLVGEDGHIK
Lys2
11.88734459
1
uM
QL-XII-47 BCWM.1 CDK4
DLKPENILVTSGGTVK
Lys2
-9.229049081
1
uM
QL-XII-47 BCWM.1 CDK7
DLKPNNLLLDENGVLK
Lys2
15.31231831
1
uM
QL-XII-47 BCWM.1 ACK
TVSVAVKCLKPDVLSQPEAMDDFIR
Lys1
16.75144083
1
uM
QL-XII-47 BCWM.1 ATR
FYIMMCKPK
ATP
0.044349501
1
uM
QL-XII-47 BCWM.1 BRAF
DLKSNNIFLHEDLTVK
Lys2
17.78977881
1
uM
QL-XII-47 BCWM.1 CaMK2g
TSTQEYAAKIINTK
Lys1
4.50076179
1
uM
QL-XII-47 BCWM.1 CDK11,CDK8
DLKPANILVMGEGPER
Lys2
14.74034939
1
uM
QL-XII-47 BCWM.1 CDK2
DLKPQNLLINTEGAIK
Lys2
-1.556399301
1
uM
QL-XII-47 BCWM.1 CDK5
DLKPQNLLINR
Lys2
4.004453656
1
uM
QL-XII-47 BCWM.1 CDK6
DLKPQNILVTSSGQIK
Lys2
-0.544166997
1
uM
QL-XII-47 BCWM.1 ABL,ARG
LMTGDTYTAHAGAKFPIK
Activation Loop
-4.884271122
1
uM
QL-XII-47 BCWM.1 ABL,ARG
YSLTVAVKTLKEDTMEVEEFLK
Lys1
23.94636209
1
uM
QL-XII-47 BCWM.1 AMPKa1,AMPKa2
DLKPENVLLDAHMNAK
Lys2
18.43323382
1
uM
QL-XII-47 BCWM.1 ARAF
DLKSNNIFLHEGLTVK
Lys2
4.534711447
1
uM
QL-XII-47 BCWM.1 AurB
SHFIVALKVLFK
Lys1
7.861261294
1
uM
QL-XII-47 BCWM.1 BARK1
DLKPANILLDEHGHVR
Lys2
-22.46332421
1
uM
QL-XII-47 BCWM.1 BTK
YVLDDEYTSSVGSKFPVR
Activation Loop
70.55327861
1
uM
QL-XII-47 BCWM.1 CAMK1D
LFAVKCIPK
Lys1
0.033712822
1
uM
QL-XII-47 BCWM.1 CDC2
DLKPQNLLIDDKGTIK
Lys2
-11.32754424
1
uM
QL-XII-47 BCWM.1 CHK2
DLKPENVLLSSQEEDCLIK
Lys2
1.250240618
1
uM
QL-XII-47 BCWM.1 CHK1
DIKPENLLLDER
Lys2
2.996204004
1
uM
  • Page 1 of 16
  • 1 to 25 of 378 records