QL-X-138 KiNativ -- single dose experiment - Dataset (ID:20204)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| QL-X-138 | BCWM.1 | RSKL1_domain1 | VLGVIDKVLLVMDTR | Protein Kinase Domain | 51.34744349 | 1 | uM |
| QL-X-138 | BCWM.1 | SGK3 | FYAVKVLQK | Lys1 | -3.700314175 | 1 | uM |
| QL-X-138 | BCWM.1 | SLK | DLKAGNILFTLDGDIK | Lys2 | -4.760224095 | 1 | uM |
| QL-X-138 | BCWM.1 | SMG1 | DTVTIHSVGGTITILPTKTKPK | ATP | -2.05694511 | 1 | uM |
| QL-X-138 | BCWM.1 | SNRK | DLKPENVVFFEK | Lys2 | 27.48203669 | 1 | uM |
| QL-X-138 | BCWM.1 | SRPK1 | IIHTDIKPENILLSVNEQYIR | Lys2 | 40.93926551 | 1 | uM |
| QL-X-138 | BCWM.1 | SRPK1/2 | FVAMKVVK | Lys1 | 16.14542611 | 1 | uM |
| QL-X-138 | BCWM.1 | STLK5 | YSVKVLPWLSPEVLQQNLQGYDAK | Activation Loop | 83.55619082 | 1 | uM |
| QL-X-138 | BCWM.1 | SYK | ISDFGLSKALR | Activation Loop | -7.149695441 | 1 | uM |
| QL-X-138 | BCWM.1 | MAP3K7,TAK1 | DLKPPNLLLVAGGTVLK | Lys2 | 80.23274866 | 1 | uM |
| QL-X-138 | BCWM.1 | TAO1,TAOK3 | DIKAGNILLTEPGQVK | Lys2 | -18.0296974 | 1 | uM |
| QL-X-138 | BCWM.1 | TAOK2 | DVKAGNILLSEPGLVK | Lys2 | 0.401729874 | 1 | uM |
| QL-X-138 | BCWM.1 | TBK1 | TGDLFAIKVFNNISFLRPVDVQMR | Lys1 | 62.64645592 | 1 | uM |
| QL-X-138 | BCWM.1 | TEC | YVLDDQYTSSSGAKFPVK | Activation Loop | >90 | 1 | uM |
| QL-X-138 | BCWM.1 | TLK1 | YLNEIKPPIIHYDLKPGNILLVDGTACGEIK | Lys2 | 41.67420927 | 1 | uM |
| QL-X-138 | BCWM.1 | TLK1/2 | YLNEIKPPIIHYDLKPGNILLVNGTACGEIK | Lys2 | 42.85258968 | 1 | uM |
| QL-X-138 | BCWM.1 | ULK1 | DLKPQNILLSNPAGR | Lys2 | -23.63664638 | 1 | uM |
| QL-X-138 | BCWM.1 | VRK2 | MLDVLEYIHENEYVHGDIKAANLLLGYK | Lys2 | 66.79689905 | 1 | uM |
| QL-X-138 | BCWM.1 | Wnk1,Wnk2,Wnk3 | DLKCDNIFITGPTGSVK | Lys2 | -23.51635392 | 1 | uM |
| QL-X-138 | BCWM.1 | ZC1/HGK,ZC2/TNIK,ZC3/MINK | DIKGQNVLLTENAEVK | Lys2 | -15.05661431 | 1 | uM |
| QL-X-138 | BCWM.1 | ZC2/TNIK | TGQLAAIKVMDVTGDEEEEIKQEINMLKK | Lys1 | 30.08512389 | 1 | uM |
| QL-X-138 | BCWM.1 | KCC2D | IPTGQEYAAKIINTKK | Lys1 | 6.541139364 | 1 | uM |
| QL-X-138 | BCWM.1 | KC1G2 | DVKPENFLVGRPGTK | Lys2 | 16.69415688 | 1 | uM |
| QL-X-138 | BCWM.1 | EPHB1 | YLQDDTSDPTYTSSLGGKIPVR | Activation Loop | 33.17017737 | 1 | uM |
| QL-X-138 | BCWM.1 | MK01 | DLKPSNLLLNTTCDLK | Lys2 | 9.89754818 | 1 | uM |