Crizotinib KINOMEscan-2 - Dataset (ID:20200)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Crizotinib | AURKB | 76.0 | nM |
Crizotinib | ABL1-nonphosphorylated | 78.0 | nM |
Crizotinib | MAP4K5 | 79.0 | nM |
Crizotinib | MAP4K2 | 80.0 | nM |
Crizotinib | TRKC | 82.0 | nM |
Crizotinib | ABL1(H396P)-phosphorylated | 87.0 | nM |
Crizotinib | TRKA | 95.0 | nM |
Crizotinib | ABL1(Q252H)-nonphosphorylated | 97.0 | nM |
Crizotinib | ABL1(M351T)-phosphorylated | 97.0 | nM |
Crizotinib | EPHA2 | 100.0 | nM |
Crizotinib | ABL1(Q252H)-phosphorylated | 100.0 | nM |
Crizotinib | TIE1 | 110.0 | nM |
Crizotinib | TNNI3K | 110.0 | nM |
Crizotinib | BLK | 110.0 | nM |
Crizotinib | MAP3K3 | 110.0 | nM |
Crizotinib | ABL1-phosphorylated | 110.0 | nM |
Crizotinib | EPHB1 | 120.0 | nM |
Crizotinib | SNARK | 120.0 | nM |
Crizotinib | EPHA1 | 140.0 | nM |
Crizotinib | CASK | 140.0 | nM |
Crizotinib | ABL1(E255K)-phosphorylated | 170.0 | nM |
Crizotinib | M3K12 | 170.0 | nM |
Crizotinib | FAK2 | 190.0 | nM |
Crizotinib | SIK2 | 200.0 | nM |
Crizotinib | JAK3(JH1domain-catalytic) | 200.0 | nM |