Crizotinib KINOMEscan-2 - Dataset (ID:20200)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Crizotinib | AAK1 | 2300.0 | nM |
| Crizotinib | ABL1(E255K)-phosphorylated | 170.0 | nM |
| Crizotinib | ABL1(F317I)-nonphosphorylated | 2700.0 | nM |
| Crizotinib | ABL1(F317I)-phosphorylated | 3200.0 | nM |
| Crizotinib | ABL1(F317L)-nonphosphorylated | 610.0 | nM |
| Crizotinib | ABL1(F317L)-phosphorylated | 590.0 | nM |
| Crizotinib | ABL1(H396P)-nonphosphorylated | 33.0 | nM |
| Crizotinib | ABL1(H396P)-phosphorylated | 87.0 | nM |
| Crizotinib | ABL1(M351T)-phosphorylated | 97.0 | nM |
| Crizotinib | ABL1(Q252H)-nonphosphorylated | 97.0 | nM |
| Crizotinib | ABL1(Q252H)-phosphorylated | 100.0 | nM |
| Crizotinib | ABL1(T315I)-nonphosphorylated | 12.0 | nM |
| Crizotinib | ABL1(T315I)-phosphorylated | 10.0 | nM |
| Crizotinib | ABL1(Y253F)-phosphorylated | 74.0 | nM |
| Crizotinib | ABL1-nonphosphorylated | 78.0 | nM |
| Crizotinib | ABL1-phosphorylated | 110.0 | nM |
| Crizotinib | ABL2 | 460.0 | nM |
| Crizotinib | ACVR1 | 440.0 | nM |
| Crizotinib | ACVR1B | 860.0 | nM |
| Crizotinib | ACVR2A | nM | |
| Crizotinib | ACVR2B | nM | |
| Crizotinib | ACVRL1 | nM | |
| Crizotinib | ADCK3 | nM | |
| Crizotinib | ADCK4 | 1100.0 | nM |
| Crizotinib | AKT1 | nM |