Crizotinib KINOMEscan-2 - Dataset (ID:20200)

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Small Molecule Protein Kd Conc unit
Crizotinib KIT
nM
Crizotinib KIT(A829P)
nM
Crizotinib KIT(D816H)
nM
Crizotinib KIT(D816V) 3700.0
nM
Crizotinib KIT(L576P)
nM
Crizotinib KIT(V559D)
nM
Crizotinib KIT(V559D,T670I) 800.0
nM
Crizotinib KIT(V559D,V654A)
nM
Crizotinib LATS1
nM
Crizotinib LATS2
nM
Crizotinib LCK 30.0
nM
Crizotinib LIMK1 830.0
nM
Crizotinib LIMK2 690.0
nM
Crizotinib LKB1
nM
Crizotinib LOK 44.0
nM
Crizotinib LRRK2
nM
Crizotinib LRRK2(G2019S)
nM
Crizotinib LTK 12.0
nM
Crizotinib LYN 940.0
nM
Crizotinib M3K13 230.0
nM
Crizotinib MAK
nM
Crizotinib MAP3K1 1100.0
nM
Crizotinib MAP3K15 2800.0
nM
Crizotinib M3K2 72.0
nM
Crizotinib MAP3K3 110.0
nM