Crizotinib KINOMEscan-2 - Dataset (ID:20200)

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Small Molecule Protein Kd Conc unit
Crizotinib FES 450.0
nM
Crizotinib FGFR1
nM
Crizotinib FGFR2
nM
Crizotinib FGFR3 2700.0
nM
Crizotinib FGFR3(G697C) 3500.0
nM
Crizotinib FGFR4
nM
Crizotinib FGR 670.0
nM
Crizotinib VGFR1 2300.0
nM
Crizotinib FLT3 850.0
nM
Crizotinib FLT3(D835H) 500.0
nM
Crizotinib FLT3(D835Y) 210.0
nM
Crizotinib FLT3(ITD) 730.0
nM
Crizotinib FLT3(K663Q) 900.0
nM
Crizotinib FLT3(N841I) 860.0
nM
Crizotinib FLT3(R834Q) 3000.0
nM
Crizotinib FLT4
nM
Crizotinib FRK 2900.0
nM
Crizotinib FYN 1300.0
nM
Crizotinib GAK
nM
Crizotinib GCN2(Kin.Dom.2,S808G)
nM
Crizotinib GRK1
nM
Crizotinib GRK4 4200.0
nM
Crizotinib GRK7
nM
Crizotinib GSK3A
nM
Crizotinib GSK3B
nM