Crizotinib KINOMEscan-2 - Dataset (ID:20200)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Crizotinib | FES | 450.0 | nM |
Crizotinib | FGFR1 | nM | |
Crizotinib | FGFR2 | nM | |
Crizotinib | FGFR3 | 2700.0 | nM |
Crizotinib | FGFR3(G697C) | 3500.0 | nM |
Crizotinib | FGFR4 | nM | |
Crizotinib | FGR | 670.0 | nM |
Crizotinib | VGFR1 | 2300.0 | nM |
Crizotinib | FLT3 | 850.0 | nM |
Crizotinib | FLT3(D835H) | 500.0 | nM |
Crizotinib | FLT3(D835Y) | 210.0 | nM |
Crizotinib | FLT3(ITD) | 730.0 | nM |
Crizotinib | FLT3(K663Q) | 900.0 | nM |
Crizotinib | FLT3(N841I) | 860.0 | nM |
Crizotinib | FLT3(R834Q) | 3000.0 | nM |
Crizotinib | FLT4 | nM | |
Crizotinib | FRK | 2900.0 | nM |
Crizotinib | FYN | 1300.0 | nM |
Crizotinib | GAK | nM | |
Crizotinib | GCN2(Kin.Dom.2,S808G) | nM | |
Crizotinib | GRK1 | nM | |
Crizotinib | GRK4 | 4200.0 | nM |
Crizotinib | GRK7 | nM | |
Crizotinib | GSK3A | nM | |
Crizotinib | GSK3B | nM |