Crizotinib KINOMEscan-2 - Dataset (ID:20200)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Crizotinib | DCAMKL2 | 370.0 | nM |
Crizotinib | DCAMKL3 | nM | |
Crizotinib | DDR1 | 510.0 | nM |
Crizotinib | DDR2 | nM | |
Crizotinib | M3K12 | 170.0 | nM |
Crizotinib | DMPK | 1400.0 | nM |
Crizotinib | DMPK2 | nM | |
Crizotinib | DRAK1 | nM | |
Crizotinib | DRAK2 | nM | |
Crizotinib | DYRK1A | nM | |
Crizotinib | DYRK1B | nM | |
Crizotinib | DYRK2 | 4000.0 | nM |
Crizotinib | EGFR | nM | |
Crizotinib | EGFR(E746-A750del) | nM | |
Crizotinib | EGFR(G719C) | 2700.0 | nM |
Crizotinib | EGFR(G719S) | nM | |
Crizotinib | EGFR(L747-E749del, A750P) | nM | |
Crizotinib | EGFR(L747-S752del, P753S) | nM | |
Crizotinib | EGFR(L747-T751del,Sins) | nM | |
Crizotinib | EGFR(L858R) | nM | |
Crizotinib | EGFR(L858R,T790M) | nM | |
Crizotinib | EGFR(L861Q) | 2700.0 | nM |
Crizotinib | EGFR(S752-I759del) | nM | |
Crizotinib | EGFR(T790M) | nM | |
Crizotinib | EIF2AK1 | nM |