TAE-684 KINOMEscan - Dataset (ID:20199)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
NVP-TAE684 | HCK | 410.0 | nM |
NVP-TAE684 | HIPK1 | 4400.0 | nM |
NVP-TAE684 | HIPK2 | 4400.0 | nM |
NVP-TAE684 | HIPK3 | 6900.0 | nM |
NVP-TAE684 | HIPK4 | 350.0 | nM |
NVP-TAE684 | M4K1 | 140.0 | nM |
NVP-TAE684 | HUNK | 350.0 | nM |
NVP-TAE684 | ICK | 4000.0 | nM |
NVP-TAE684 | IGF1R | 2.7 | nM |
NVP-TAE684 | IKKA | nM | |
NVP-TAE684 | IKKB | nM | |
NVP-TAE684 | IKKE | 1100.0 | nM |
NVP-TAE684 | INSR | 2.4 | nM |
NVP-TAE684 | INSRR | 6.2 | nM |
NVP-TAE684 | IRAK1 | 45.0 | nM |
NVP-TAE684 | IRAK3 | 160.0 | nM |
NVP-TAE684 | IRAK4 | 77.0 | nM |
NVP-TAE684 | ITK | 34.0 | nM |
NVP-TAE684 | JAK1(JH1domain-catalytic) | 410.0 | nM |
NVP-TAE684 | JAK1(JH2domain-pseudokinase) | 300.0 | nM |
NVP-TAE684 | JAK2(JH1domain-catalytic) | 16.0 | nM |
NVP-TAE684 | JAK3(JH1domain-catalytic) | 17.0 | nM |
NVP-TAE684 | JNK1 | 160.0 | nM |
NVP-TAE684 | MK09 | 280.0 | nM |
NVP-TAE684 | JNK3 | 67.0 | nM |