TAE-684 KINOMEscan - Dataset (ID:20199)

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Small Molecule Protein Kd Conc unit
NVP-TAE684 HCK 410.0
nM
NVP-TAE684 HIPK1 4400.0
nM
NVP-TAE684 HIPK2 4400.0
nM
NVP-TAE684 HIPK3 6900.0
nM
NVP-TAE684 HIPK4 350.0
nM
NVP-TAE684 M4K1 140.0
nM
NVP-TAE684 HUNK 350.0
nM
NVP-TAE684 ICK 4000.0
nM
NVP-TAE684 IGF1R 2.7
nM
NVP-TAE684 IKKA
nM
NVP-TAE684 IKKB
nM
NVP-TAE684 IKKE 1100.0
nM
NVP-TAE684 INSR 2.4
nM
NVP-TAE684 INSRR 6.2
nM
NVP-TAE684 IRAK1 45.0
nM
NVP-TAE684 IRAK3 160.0
nM
NVP-TAE684 IRAK4 77.0
nM
NVP-TAE684 ITK 34.0
nM
NVP-TAE684 JAK1(JH1domain-catalytic) 410.0
nM
NVP-TAE684 JAK1(JH2domain-pseudokinase) 300.0
nM
NVP-TAE684 JAK2(JH1domain-catalytic) 16.0
nM
NVP-TAE684 JAK3(JH1domain-catalytic) 17.0
nM
NVP-TAE684 JNK1 160.0
nM
NVP-TAE684 MK09 280.0
nM
NVP-TAE684 JNK3 67.0
nM