TAE-684 KINOMEscan - Dataset (ID:20199)
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| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| NVP-TAE684 | IKKB | nM | |
| NVP-TAE684 | IKKE | 1100.0 | nM |
| NVP-TAE684 | INSR | 2.4 | nM |
| NVP-TAE684 | INSRR | 6.2 | nM |
| NVP-TAE684 | IRAK1 | 45.0 | nM |
| NVP-TAE684 | IRAK3 | 160.0 | nM |
| NVP-TAE684 | IRAK4 | 77.0 | nM |
| NVP-TAE684 | ITK | 34.0 | nM |
| NVP-TAE684 | JAK1(JH1domain-catalytic) | 410.0 | nM |
| NVP-TAE684 | JAK1(JH2domain-pseudokinase) | 300.0 | nM |
| NVP-TAE684 | JAK2(JH1domain-catalytic) | 16.0 | nM |
| NVP-TAE684 | JAK3(JH1domain-catalytic) | 17.0 | nM |
| NVP-TAE684 | JNK1 | 160.0 | nM |
| NVP-TAE684 | JNK3 | 67.0 | nM |
| NVP-TAE684 | KC1G1 | nM | |
| NVP-TAE684 | KC1G2 | nM | |
| NVP-TAE684 | KCC2D | 570.0 | nM |
| NVP-TAE684 | KCC4 | 30.0 | nM |
| NVP-TAE684 | KGP1 | 430.0 | nM |
| NVP-TAE684 | KGP2 | 240.0 | nM |
| NVP-TAE684 | KIT | 110.0 | nM |
| NVP-TAE684 | KIT(A829P) | 220.0 | nM |
| NVP-TAE684 | KIT(D816H) | 140.0 | nM |
| NVP-TAE684 | KIT(D816V) | 26.0 | nM |
| NVP-TAE684 | KIT(L576P) | 49.0 | nM |