TAE-684 KINOMEscan - Dataset (ID:20199)

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Small Molecule Protein Kd Conc unit
NVP-TAE684 AKT2
nM
NVP-TAE684 AKT3
nM
NVP-TAE684 ALK 1.1
nM
NVP-TAE684 AMPK-alpha1 27.0
nM
NVP-TAE684 AMPK-alpha2 49.0
nM
NVP-TAE684 ANKK1 9400.0
nM
NVP-TAE684 AURKA 44.0
nM
NVP-TAE684 AURKB 150.0
nM
NVP-TAE684 AURKC 33.0
nM
NVP-TAE684 AXL 12.0
nM
NVP-TAE684 BIKE 1900.0
nM
NVP-TAE684 BLK 130.0
nM
NVP-TAE684 BMPR1A 170.0
nM
NVP-TAE684 BMPR1B 0.9
nM
NVP-TAE684 BMPR2 3900.0
nM
NVP-TAE684 BMX 1100.0
nM
NVP-TAE684 BRAF
nM
NVP-TAE684 BRAF(V600E)
nM
NVP-TAE684 BRSK1 310.0
nM
NVP-TAE684 BRSK2 190.0
nM
NVP-TAE684 BTK 23.0
nM
NVP-TAE684 CAMK1 1100.0
nM
NVP-TAE684 CAMK1D 230.0
nM
NVP-TAE684 CAMK1G 3000.0
nM
NVP-TAE684 CAMK2A 980.0
nM