TAE-684 KINOMEscan - Dataset (ID:20199)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| NVP-TAE684 | INSRR | 6.2 | nM |
| NVP-TAE684 | EGFR(T790M) | 7.1 | nM |
| NVP-TAE684 | FLT3(K663Q) | 8.2 | nM |
| NVP-TAE684 | FLT3(ITD) | 8.6 | nM |
| NVP-TAE684 | ULK3 | 11.0 | nM |
| NVP-TAE684 | FLT3(N841I) | 11.0 | nM |
| NVP-TAE684 | CAMKK2 | 11.0 | nM |
| NVP-TAE684 | CLK1 | 12.0 | nM |
| NVP-TAE684 | MARK3 | 12.0 | nM |
| NVP-TAE684 | MARK4 | 12.0 | nM |
| NVP-TAE684 | AXL | 12.0 | nM |
| NVP-TAE684 | YANK1 | 13.0 | nM |
| NVP-TAE684 | PHKG2 | 13.0 | nM |
| NVP-TAE684 | NUAK1 | 13.0 | nM |
| NVP-TAE684 | DCAMKL3 | 14.0 | nM |
| NVP-TAE684 | ABL1(F317I)-phosphorylated | 14.0 | nM |
| NVP-TAE684 | TIE1 | 15.0 | nM |
| NVP-TAE684 | SIK1 | 15.0 | nM |
| NVP-TAE684 | FLT3 | 15.0 | nM |
| NVP-TAE684 | JAK2(JH1domain-catalytic) | 16.0 | nM |
| NVP-TAE684 | DCAMKL2 | 16.0 | nM |
| NVP-TAE684 | JAK3(JH1domain-catalytic) | 17.0 | nM |
| NVP-TAE684 | SIK2 | 17.0 | nM |
| NVP-TAE684 | PHKG1 | 17.0 | nM |
| NVP-TAE684 | RSK2(Kin.Dom.1-N-terminal) | 17.0 | nM |