TAE-684 KINOMEscan - Dataset (ID:20199)
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| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| NVP-TAE684 | ROS1 | 0.5 | nM |
| NVP-TAE684 | ULK1 | 0.8 | nM |
| NVP-TAE684 | LRRK2(G2019S) | 0.9 | nM |
| NVP-TAE684 | BMPR1B | 0.9 | nM |
| NVP-TAE684 | PLK4 | 0.9 | nM |
| NVP-TAE684 | LTK | 1.0 | nM |
| NVP-TAE684 | FAK2 | 1.1 | nM |
| NVP-TAE684 | ALK | 1.1 | nM |
| NVP-TAE684 | FAK1 | 1.1 | nM |
| NVP-TAE684 | SNARK | 1.2 | nM |
| NVP-TAE684 | LRRK2 | 1.4 | nM |
| NVP-TAE684 | FER | 1.4 | nM |
| NVP-TAE684 | TNK1 | 1.8 | nM |
| NVP-TAE684 | ULK2 | 1.8 | nM |
| NVP-TAE684 | TNK2 | 2.0 | nM |
| NVP-TAE684 | FLT3(D835Y) | 2.0 | nM |
| NVP-TAE684 | INSR | 2.4 | nM |
| NVP-TAE684 | IGF1R | 2.7 | nM |
| NVP-TAE684 | STK33 | 3.2 | nM |
| NVP-TAE684 | EGFR(L858R,T790M) | 3.4 | nM |
| NVP-TAE684 | FES | 4.8 | nM |
| NVP-TAE684 | FLT3(D835H) | 4.9 | nM |
| NVP-TAE684 | DCLK1 | 4.9 | nM |
| NVP-TAE684 | GAK | 5.3 | nM |
| NVP-TAE684 | ABL1(T315I)-phosphorylated | 5.4 | nM |